SCHEMBL20344786

SCHEMBL20344786

COC(=O)Cc1c(C)cn2cc(-c3cccc(Cl)c3)nc2c1-c1cc2c(cc1OC(C)(C)C)OCCC2

nearest known ligand 0.35

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 2/20 0.33
THRB P10828 1/20 0.33
EPHB4 P54760 3/20 0.31
PDE4B Q07343 1/20 0.31
MAPT P10636 1/20 0.31
MAPK1 P28482 1/20 0.31
P2RX3 P56373 1/20 0.31
TRPV1 Q8NER1 1/20 0.31
CNR2 P34972 1/20 0.31
AVPR1B P47901 3/20 0.30
WDR5 P61964 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL20344807 0.90 P2RX7 (0.33) P2RX7
SCHEMBL17039255 0.81 CLK1 (0.40) MAPTMAPK1P2RX3
SCHEMBL17039306 0.78 FABP4 (0.35) P2RX7MAPT
SCHEMBL17039251 0.74 P2RX3 (0.36) P2RX3AVPR1B
SCHEMBL17029066 0.74 P2RX3 (0.36) P2RX3AVPR1B
SCHEMBL17029065 0.74 P2RX3 (0.36) P2RX3AVPR1B
SCHEMBL17039259 0.74 NR1I2 (0.39) PDE4BMAPTMAPK1AVPR1B
SCHEMBL17039247 0.73 KDM4E (0.40) THRBMAPTCNR2
SCHEMBL17029018 0.73 NR1I2 (0.40)
SCHEMBL18364987 0.73 CLK1 (0.35) P2RX3TRPV1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3107913-B1 INHIBITORS OF HUMAN IMMUNODEFICIENCY VIRUS REPLICATION VIIV HEALTHCARE UK NO 5 LTD (GB) 2018-07-04 EP disclosed