SCHEMBL17059172

SCHEMBL17059172

Cc1nnc(C2(c3ccccc3)CC2)c(N)n1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
OPRM1 P35372 3/20 0.38
ADORA2A P29274 2/20 0.38
DRD4 P21917 1/20 0.38
PIK3CD O00329 7/20 0.37
PIK3R1 P27986 7/20 0.37
GRIN2D O15399 1/20 0.37
GRIN3B O60391 1/20 0.37
CHRM2 P08172 1/20 0.37
CHRM1 P11229 1/20 0.37
GRIN1 Q05586 1/20 0.37
KCNH2 Q12809 1/20 0.37
GRIN2A Q12879 1/20 0.37
GRIN2B Q13224 1/20 0.37
GRIN2C Q14957 1/20 0.37
GRIN3A Q8TCU5 1/20 0.37
CYP2D6 P10635 1/20 0.37
COMT P21964 1/20 0.35
CHEK1 O14757 1/20 0.34
ABL1 P00519 1/20 0.34
PDGFRB P09619 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL9607818 0.83 CSNK1A1 (0.44) OPRM1ADORA2ADRD4PIK3CDPIK3R1
SCHEMBL9607809 0.79 CSNK1A1 (0.43) OPRM1ADORA2ADRD4CLK4MEN1
SCHEMBL9607808 0.77 CSNK1A1 (0.42) ADORA2ACLK4MEN1KMT2AHSD11B1
SCHEMBL17059348 0.73 ALDH1A1 (0.38) MEN1KMT2AHSD11B1
SCHEMBL9607812 0.70 HSD11B1 (0.41) BACE1MEN1KMT2AHSD11B1
SCHEMBL9607820 0.69 ALDH1A1 (0.43) BACE1MEN1KMT2AHSD11B1
SCHEMBL976986 0.68 BACE1 (0.46) ADORA2AGSK3BPIK3CGBACE1HSD11B1
SCHEMBL2256573 0.65 OPRM1 (0.67) OPRM1DRD4GRIN2DGRIN3BCHRM2
SCHEMBL2256575 0.65 OPRM1 (0.67) OPRM1DRD4GRIN2DGRIN3BCHRM2
SCHEMBL2658676 0.65 CLK4 (0.66) OPRM1ADORA2ACYP2D6CHEK1ABL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2451807-B1 CYCLIC TRIAZO SODIUM CHANNEL BLOCKERS UNIV GREENWICH (GB) 2015-09-02 EP disclosed