SCHEMBL1707751

SCHEMBL1707751

COC(=O)/C=C/c1cnc(N[C@@H]2CCCN(CCc3cccc(F)c3)C2)cn1

nearest known ligand 0.42

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
SLC6A3 Q01959 1/20 0.41
MAPK1 P28482 1/20 0.39
CCR3 P51677 1/20 0.39
ATM Q13315 1/20 0.39
CCNT1 O60563 1/20 0.38
HTR2A P28223 1/20 0.38
ALDH1A1 P00352 2/20 0.37
KDM4E B2RXH2 1/20 0.37
HPGD P15428 1/20 0.37
KAT2B Q92831 1/20 0.37
CACNA1G O43497 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1706845 0.95 ATM (0.40) SLC6A3ATMCCNT1HTR2ACACNA1G
SCHEMBL1706846 0.95 ATM (0.40) SLC6A3ATMCCNT1HTR2ACACNA1G
SCHEMBL1706817 0.91 SLC6A3 (0.43) SLC6A3MAPK1CCR3ATMCCNT1
SCHEMBL1706819 0.91 SLC6A3 (0.43) SLC6A3MAPK1CCR3ATMCCNT1
SCHEMBL1707102 0.89 SLC6A3 (0.41) SLC6A3MAPK1CCR3ATMHTR2A
SCHEMBL1707095 0.89 SLC6A3 (0.41) SLC6A3MAPK1CCR3ATMHTR2A
SCHEMBL1707646 0.89 ROCK2 (0.40) MAPK1CCR3ALDH1A1KDM4EKAT2B
Hydrochloric Acid SCHEMBL1706803 0.89 SLC6A3 (0.41) SLC6A3MAPK1CCR3ATMHTR2A
Hydrochloric Acid SCHEMBL1707440 0.89 SLC6A3 (0.41) SLC6A3MAPK1CCR3ATMHTR2A
Hydrochloric Acid SCHEMBL1706805 0.89 SLC6A3 (0.41) SLC6A3MAPK1CCR3ATMHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1981877-B1 N-HYDROXYACRYLAMIDE COMPOUNDS ASTELLAS PHARMA INC (JP) 2012-04-18 EP disclosed