SCHEMBL1708026

SCHEMBL1708026

CCc1nc2ccc(F)cc2n1-c1cccc(CNc2ccc3c(c2)OC(C)[C@H]3OC(C)=O)c1C

nearest known ligand 0.34

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
BMI1 P35226 3/20 0.33
HDAC6 Q9UBN7 1/20 0.32
NPC1 O15118 2/20 0.31
RAB9A P51151 2/20 0.31
PDE2A O00408 2/20 0.31
NTRK1 P04629 1/20 0.31
NTRK2 Q16620 1/20 0.31
MAPT P10636 3/20 0.30
KDM4E B2RXH2 2/20 0.30
MEN1 O00255 1/20 0.30
ALDH1A1 P00352 1/20 0.30
GAA P10253 1/20 0.30
KMT2A Q03164 1/20 0.30
HSD17B10 Q99714 1/20 0.30
TDP1 Q9NUW8 1/20 0.30
GPR55 Q9Y2T6 1/20 0.30
L3MBTL1 Q9Y468 1/20 0.30
TP53 P04637 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708080 0.93 NPC1 (0.35) BMI1NPC1RAB9APDE2AMAPT
SCHEMBL1707997 0.91 PDE2A (0.33) NPC1RAB9APDE2ANTRK1NTRK2
SCHEMBL1708155 0.91 NTRK1 (0.37) NPC1RAB9ANTRK1NTRK2MAPT
SCHEMBL1708298 0.91 PDE10A (0.33) NPC1RAB9APDE2AMAPTKDM4E
SCHEMBL1708150 0.87 NPC1 (0.39) NPC1RAB9AMAPTKDM4EMEN1
SCHEMBL1708438 0.86 GFER (0.38) NPC1RAB9AMAPTKDM4EMEN1
SCHEMBL1708134 0.86 INSR (0.30) NPC1RAB9ANTRK1NTRK2GAA
SCHEMBL1707879 0.85 MAPT (0.34) BMI1HDAC6NPC1RAB9APDE2A
SCHEMBL1708106 0.85 NPC1 (0.35) NPC1RAB9AMAPTKDM4EMEN1
SCHEMBL1708122 0.85 MAPT (0.33) BMI1HDAC6NPC1RAB9APDE2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed