SCHEMBL1707997

SCHEMBL1707997

CCc1nc2ccc(Cl)cc2n1-c1cccc(CNc2ccc3c(c2)OC(C)[C@H]3OC(C)=O)c1C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PDE2A O00408 3/20 0.33
SMN1; SMN2 Q16637 2/20 0.31
HTT P42858 1/20 0.31
MAPT P10636 6/20 0.31
TP53 P04637 4/20 0.31
ALDH1A1 P00352 1/20 0.31
PKM P14618 1/20 0.31
IDH1 O75874 1/20 0.31
NTRK1 P04629 2/20 0.31
NTRK2 Q16620 2/20 0.31
SETDB1 Q15047 1/20 0.31
MEN1 O00255 1/20 0.31
KMT2A Q03164 1/20 0.31
THRB P10828 1/20 0.31
NPSR1 Q6W5P4 1/20 0.30
POLB P06746 1/20 0.30
ACSS2 Q9NR19 1/20 0.30
LMNA P02545 2/20 0.30
NPC1 O15118 1/20 0.30
MAPK1 P28482 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708026 0.91 BMI1 (0.33) PDE2AMAPTTP53ALDH1A1NTRK1
SCHEMBL1708155 0.91 NTRK1 (0.37) SMN1; SMN2HTTMAPTTP53ALDH1A1
SCHEMBL1708438 0.86 GFER (0.38) SMN1; SMN2MAPTTP53ALDH1A1MEN1
SCHEMBL1708134 0.86 INSR (0.30) NTRK1NTRK2THRBNPC1RAB9A
SCHEMBL1708250 0.85 ALDH1A1 (0.34) PDE2AMAPTALDH1A1PKMIDH1
SCHEMBL1708106 0.85 NPC1 (0.35) SMN1; SMN2HTTMAPTTP53ALDH1A1
SCHEMBL1708264 0.85 ALDH1A1 (0.34) PDE2AMAPTALDH1A1PKMIDH1
SCHEMBL1708631 0.85 NPC1 (0.35) SMN1; SMN2HTTMAPTTP53ALDH1A1
SCHEMBL1708080 0.84 NPC1 (0.35) PDE2ASMN1; SMN2MAPTTP53ALDH1A1
SCHEMBL1708139 0.83 GFER (0.39) PDE2ASMN1; SMN2MAPTTP53ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed