SCHEMBL1708145

SCHEMBL1708145

CC(=O)O[C@H]1c2ccc(NCc3cccc(-n4c(C5CC5)nc5ccccc54)c3C)cc2OC1C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TSHR P16473 3/20 0.33
NTRK1 P04629 1/20 0.33
NTRK2 Q16620 1/20 0.33
MAPK1 P28482 1/20 0.33
BMI1 P35226 1/20 0.33
ALDH1A1 P00352 3/20 0.32
LMNA P02545 2/20 0.32
NPSR1 Q6W5P4 2/20 0.32
MAPT P10636 5/20 0.32
L3MBTL1 Q9Y468 4/20 0.32
CHEK1 O14757 1/20 0.32
ATR Q13535 1/20 0.32
PDCD1 Q15116 1/20 0.32
ATRIP Q8WXE1 1/20 0.32
CD274 Q9NZQ7 1/20 0.32
INSR P06213 1/20 0.31
IGF1R P08069 1/20 0.31
GAA P10253 4/20 0.31
RAB9A P51151 2/20 0.31
NPC1 O15118 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708637 0.91 HPGD (0.37) TSHRBMI1ALDH1A1LMNAMAPT
SCHEMBL1708155 0.89 NTRK1 (0.37) TSHRNTRK1NTRK2MAPK1ALDH1A1
SCHEMBL1708162 0.88 MAPT (0.34) TSHRNTRK1NTRK2MAPK1ALDH1A1
SCHEMBL1708072 0.87 LMNA (0.37) TSHRNTRK1NTRK2MAPK1ALDH1A1
SCHEMBL1708111 0.87 NPC1 (0.33) TSHRNTRK1NTRK2MAPK1ALDH1A1
SCHEMBL1708613 0.87 ALDH1A1 (0.34) TSHRNTRK1NTRK2MAPK1ALDH1A1
SCHEMBL1708631 0.87 NPC1 (0.35) TSHRNTRK1NTRK2MAPK1ALDH1A1
SCHEMBL1708106 0.83 NPC1 (0.35) TSHRMAPK1ALDH1A1LMNAMAPT
SCHEMBL1708634 0.83 TP53 (0.35) TSHRNTRK1NTRK2MAPK1ALDH1A1
SCHEMBL1708093 0.83 NPC1 (0.38) ALDH1A1LMNAMAPTGAARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed