SCHEMBL1708111

SCHEMBL1708111

CCOc1nc2ccccc2n1-c1cccc(CNc2ccc3c(c2)OC(C)[C@H]3OC(C)=O)c1C

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 3/20 0.33
RAB9A P51151 3/20 0.33
MAPT P10636 8/20 0.33
NTRK1 P04629 2/20 0.33
NTRK2 Q16620 2/20 0.33
GAA P10253 3/20 0.33
L3MBTL1 Q9Y468 3/20 0.32
TDP1 Q9NUW8 2/20 0.32
KDM4E B2RXH2 2/20 0.32
GPR55 Q9Y2T6 1/20 0.32
ALDH1A1 P00352 3/20 0.32
LMNA P02545 1/20 0.32
MEN1 O00255 2/20 0.31
KMT2A Q03164 2/20 0.31
NPSR1 Q6W5P4 1/20 0.31
TSHR P16473 1/20 0.31
MAPK1 P28482 1/20 0.31
TP53 P04637 2/20 0.31
THRB P10828 1/20 0.31
HSD17B10 Q99714 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1708162 0.93 MAPT (0.34) NPC1RAB9AMAPTNTRK1NTRK2
SCHEMBL1708298 0.92 PDE10A (0.33) NPC1RAB9AMAPTGAAL3MBTL1
SCHEMBL1708148 0.91 MTNR1A (0.41) MAPTGAAL3MBTL1TDP1KDM4E
SCHEMBL1708155 0.90 NTRK1 (0.37) NPC1RAB9AMAPTNTRK1NTRK2
SCHEMBL1708072 0.87 LMNA (0.37) NPC1RAB9AMAPTNTRK1NTRK2
SCHEMBL1708145 0.87 TSHR (0.33) NPC1RAB9AMAPTNTRK1NTRK2
SCHEMBL1708631 0.87 NPC1 (0.35) NPC1RAB9AMAPTNTRK1NTRK2
SCHEMBL1708613 0.87 ALDH1A1 (0.34) NPC1RAB9AMAPTNTRK1NTRK2
SCHEMBL1708014 0.85 MAPT (0.35) NPC1RAB9AMAPTNTRK1NTRK2
SCHEMBL1708106 0.83 NPC1 (0.35) NPC1RAB9AMAPTGAAL3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2440541-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF Takeda Pharmaceutical Company Limited (JP) 2012-04-18 EP disclosed
WO-2010143733-A1 NOVEL FUSED CYCLIC COMPOUND AND USE THEREOF TAKEDA PHARMACEUTICAL COMPANY LIMITED (JP) 2010-12-16 WO disclosed