SCHEMBL17090002

SCHEMBL17090002

CC(C)(C)NC(=O)c1ccc(NC[C@H]2CC[C@H](NS(=O)(=O)C(C)(C)C)CC2)cc1

nearest known ligand 0.40

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
KDM1A O60341 1/20 0.40
LMNA P02545 1/20 0.40
HTT P42858 1/20 0.40
CACNA1H O95180 2/20 0.39
NPY5R Q15761 1/20 0.39
CRHR1 P34998 3/20 0.39
MAPK14 Q16539 3/20 0.36
HSPB1 P04792 1/20 0.36
CYP2C9 P11712 1/20 0.36
MAPK11 Q15759 1/20 0.36
CNR1 P21554 1/20 0.36
CNR2 P34972 1/20 0.36
CA2 P00918 1/20 0.36
USP2 O75604 1/20 0.36
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36
POLB P06746 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17090128 0.87 MEN1 (0.43) LMNANPY5RCRHR1CNR1CNR2
SCHEMBL13565746 0.87 MEN1 (0.43) LMNANPY5RCRHR1CNR1CNR2
SCHEMBL13438995 0.87 MAPK14 (0.46) NPY5RCRHR1MAPK14CNR1CNR2
SCHEMBL17090170 0.87 KDM1A (0.39) KDM1ALMNAHTTCACNA1HNPY5R
SCHEMBL11935305 0.87 MAPK14 (0.46) NPY5RCRHR1MAPK14CNR1CNR2
SCHEMBL11935324 0.86 LMNA (0.53) LMNACRHR1MAPK14HSPB1CYP2C9
SCHEMBL17090231 0.86 LMNA (0.53) LMNACRHR1MAPK14HSPB1CYP2C9
SCHEMBL17090516 0.85 CRHR1 (0.47) LMNANPY5RCRHR1MAPK14MAPK11
SCHEMBL17090363 0.84 HTT (0.44) HTTNPY5RCRHR1MAPK14POLB
SCHEMBL13565142 0.83 NPY5R (0.42) NPY5RCRHR1CNR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed