SCHEMBL17090358

SCHEMBL17090358

CC(C)(C)S(=O)(=O)N[C@H]1CC[C@H](CNc2ccc(-c3ccno3)cc2)CC1

nearest known ligand 0.39

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TOP1 P11387 1/20 0.39
CNR2 P34972 2/20 0.36
MAPK14 Q16539 1/20 0.36
NPY5R Q15761 1/20 0.35
KCNJ1 P48048 2/20 0.35
PTGS2 P35354 2/20 0.34
SYK P43405 1/20 0.34
ALDH1A1 P00352 1/20 0.33
ALDH3A1 P30838 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13565095 1.00 TOP1 (0.39) TOP1CNR2MAPK14NPY5RKCNJ1
SCHEMBL17090035 0.85 TOP1 (0.39) TOP1
SCHEMBL13564942 0.85 TOP1 (0.39) TOP1
SCHEMBL17090368 0.82 IMPDH2 (0.42) NPY5RKCNJ1SYKALDH1A1
SCHEMBL17090361 0.82 TAAR1 (0.37) CNR2MAPK14ALDH1A1ALDH3A1
SCHEMBL13565104 0.82 TAAR1 (0.37) CNR2MAPK14ALDH1A1ALDH3A1
SCHEMBL13565131 0.81 CRHR1 (0.39) CNR2ALDH1A1ALDH3A1
SCHEMBL17090321 0.81 CRHR1 (0.39) CNR2ALDH1A1ALDH3A1
SCHEMBL13565614 0.81 CRHR1 (0.39) CNR2ALDH1A1ALDH3A1
SCHEMBL17089998 0.81 CRHR1 (0.39) CNR2ALDH1A1ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9139518-B2 Amine derivative having NPY Y5 receptor antagonistic activity SHIONOGI & CO., LTD. (JP) 2015-09-22 US disclosed