SCHEMBL1709212

SCHEMBL1709212

CCN(CC1CC12CCN(Cc1ccccc1)CC2)c1cccc(C)c1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 2/20 0.45
BACE1 P56817 2/20 0.42
SCN9A Q15858 1/20 0.41
CHRM2 P08172 2/20 0.41
CHRM3 P20309 2/20 0.41
SIGMAR1 Q99720 3/20 0.40
LMNA P02545 2/20 0.39
POLB P06746 1/20 0.39
ALDH1A1 P00352 3/20 0.39
MAPT P10636 2/20 0.39
MAPK1 P28482 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
GAA P10253 1/20 0.39
BCHE P06276 1/20 0.39
KDM4E B2RXH2 2/20 0.38
CHRM1 P11229 1/20 0.38
MCL1 Q07820 1/20 0.38
OPRM1 P35372 1/20 0.38
KCNH2 Q12809 1/20 0.38
DCUN1D1 Q96GG9 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709216 0.84 ACHE (0.47) ACHESCN9ACHRM2CHRM3SIGMAR1
SCHEMBL1709211 0.70 SCN9A (0.59) ACHEBACE1SCN9ASIGMAR1LMNA
SCHEMBL1709213 0.70 SCN9A (0.58) ACHEBACE1SCN9ASIGMAR1LMNA
SCHEMBL10071963 0.68 SCN9A (0.56) ACHEBACE1SCN9ASIGMAR1LMNA
SCHEMBL1224833 0.68 TSHR (0.70) ALDH1A1TDP1
Hydrochloric Acid SCHEMBL9310741 0.67 BACE1 (0.54) ACHEBACE1CHRM2CHRM3SIGMAR1
Hydrochloric Acid SCHEMBL9310735 0.67 BACE1 (0.54) ACHEBACE1CHRM2CHRM3SIGMAR1
SCHEMBL4832242 0.66 CHRM2 (0.56) ACHEBACE1CHRM2CHRM3SIGMAR1
SCHEMBL3894897 0.66 OPRL1 (0.73) CHRM2CHRM3SIGMAR1POLBALDH1A1
SCHEMBL12203 0.66 CHRM2 (0.55) ACHEBACE1CHRM2CHRM3LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed