SCHEMBL10071963

SCHEMBL10071963

CCc1cccc(NCC2CC23CCN(Cc2ccccc2)CC3)c1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.56
NAMPT P43490 2/20 0.44
ACHE P22303 2/20 0.43
BACE1 P56817 2/20 0.43
ALDH1A1 P00352 2/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CYP3A4 P08684 1/20 0.40
HSD17B10 Q99714 1/20 0.40
FAAH O00519 1/20 0.40
SIGMAR1 Q99720 1/20 0.39
KCNH2 Q12809 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
HTT P42858 1/20 0.39
MEN1 O00255 1/20 0.39
KMT2A Q03164 1/20 0.39
OPRL1 P41146 1/20 0.39
ICMT O60725 1/20 0.39
NPFFR1 Q9GZQ6 1/20 0.38
NPFFR2 Q9Y5X5 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10072406 0.90 SCN9A (0.57) SCN9ANAMPTACHEBACE1ALDH1A1
SCHEMBL1709213 0.84 SCN9A (0.58) SCN9ANAMPTACHEBACE1ALDH1A1
SCHEMBL10071962 0.78 SCN9A (0.57) SCN9ANAMPTACHEBACE1CYP3A4
SCHEMBL1709211 0.75 SCN9A (0.59) SCN9ANAMPTACHEBACE1SIGMAR1
SCHEMBL18860348 0.73 NAMPT (0.48) SCN9ANAMPTSMN1; SMN2SIGMAR1KCNH2
SCHEMBL1709247 0.73 SCN9A (0.64) SCN9ANAMPTALDH1A1SMN1; SMN2CYP3A4
SCHEMBL1709232 0.72 SCN9A (1.00) SCN9ANAMPTACHEBACE1ALDH1A1
SCHEMBL1709234 0.72 SCN9A (0.60) SCN9ANAMPTACHEBACE1ALDH1A1
SCHEMBL9566388 0.69 CXCR4 (0.53) SCN9ANAMPTACHEBACE1CYP3A4
SCHEMBL1709212 0.68 ACHE (0.45) SCN9AACHEBACE1ALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed