SCHEMBL1709216

SCHEMBL1709216

CCN(CC1CC12CCN(Cc1ccccc1)CC2)c1ccc(Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACHE P22303 1/20 0.47
CCR3 P51677 1/20 0.46
SIGMAR1 Q99720 2/20 0.46
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 2/20 0.45
MAPT P10636 1/20 0.45
MAPK1 P28482 1/20 0.45
MCL1 Q07820 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
MEN1 O00255 2/20 0.44
KMT2A Q03164 2/20 0.44
GFER P55789 1/20 0.44
SCN9A Q15858 1/20 0.43
DRD4 P21917 2/20 0.42
CHRM2 P08172 1/20 0.42
CHRM3 P20309 1/20 0.42
DRD2 P14416 1/20 0.42
DRD3 P35462 1/20 0.42
SMN1; SMN2 Q16637 1/20 0.41
CXCR3 P49682 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709212 0.84 ACHE (0.45) ACHESIGMAR1ALDH1A1KDM4EMAPT
SCHEMBL654066 0.67 CCR3 (0.68) CCR3SIGMAR1ALDH1A1DRD4DRD2
SCHEMBL11353029 0.66 ALDH1A1 (0.83) ACHESIGMAR1ALDH1A1KDM4EMAPT
SCHEMBL16984334 0.65 ACHE (0.51) ACHESIGMAR1ALDH1A1MEN1KMT2A
SCHEMBL9566402 0.65 OPRL1 (0.48) SIGMAR1ALDH1A1MEN1KMT2ASCN9A
SCHEMBL1709249 0.64 DRD4 (0.60) SIGMAR1ALDH1A1KDM4ESCN9ADRD4
SCHEMBL653218 0.64 CCR3 (1.00) CCR3SIGMAR1KDM4EMEN1KMT2A
SCHEMBL654214 0.64 CCR3 (0.68) CCR3SIGMAR1ALDH1A1DRD4DRD2
SCHEMBL8804601 0.64 ALDH1A1 (0.67) ACHEALDH1A1KDM4EMAPTMAPK1
SCHEMBL12013906 0.63 SIGMAR1 (0.65) ACHECCR3SIGMAR1ALDH1A1MEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed