SCHEMBL1709213

SCHEMBL1709213

Cc1cc(C)cc(NCC2CC23CCN(Cc2ccccc2)CC3)c1

nearest known ligand 0.58

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 2/20 0.58
NAMPT P43490 2/20 0.46
LMNA P02545 1/20 0.43
POLB P06746 1/20 0.43
ACHE P22303 5/20 0.42
BACE1 P56817 4/20 0.42
CYP3A4 P08684 1/20 0.42
HSD17B10 Q99714 1/20 0.42
SIGMAR1 Q99720 3/20 0.41
DCUN1D1 Q96GG9 1/20 0.41
KDM4E B2RXH2 1/20 0.41
ALDH1A1 P00352 1/20 0.41
MAPT P10636 1/20 0.41
RAB9A P51151 1/20 0.41
OPRL1 P41146 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10071963 0.84 SCN9A (0.56) SCN9ANAMPTLMNAACHEBACE1
SCHEMBL10072406 0.82 SCN9A (0.57) SCN9ANAMPTPOLBACHEBACE1
SCHEMBL1709211 0.81 SCN9A (0.59) SCN9ANAMPTLMNAPOLBACHE
SCHEMBL10071962 0.80 SCN9A (0.57) SCN9ANAMPTACHEBACE1CYP3A4
SCHEMBL18860348 0.77 NAMPT (0.48) SCN9ANAMPTSIGMAR1
SCHEMBL1709232 0.74 SCN9A (1.00) SCN9ANAMPTPOLBACHEBACE1
SCHEMBL1709247 0.72 SCN9A (0.64) SCN9ANAMPTCYP3A4SIGMAR1ALDH1A1
SCHEMBL1709234 0.71 SCN9A (0.60) SCN9ANAMPTACHEBACE1CYP3A4
SCHEMBL7296842 0.70 ACHE (0.60) LMNAPOLBACHEBACE1SIGMAR1
SCHEMBL29423996 0.70 CHRM4 (0.52) SCN9AACHECYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed