SCHEMBL1709211

SCHEMBL1709211

Cc1ccc(F)c(NCC2CC23CCN(Cc2ccccc2)CC3)c1

nearest known ligand 0.59

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 1/20 0.59
SIGMAR1 Q99720 2/20 0.43
NAMPT P43490 1/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
LMNA P02545 1/20 0.42
POLB P06746 1/20 0.42
HTT P42858 1/20 0.42
ACHE P22303 3/20 0.40
BACE1 P56817 3/20 0.40
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
THRB P10828 1/20 0.40
TSHR P16473 1/20 0.39
CXCR4 P61073 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1709213 0.81 SCN9A (0.58) SCN9ASIGMAR1NAMPTKDM4ELMNA
SCHEMBL10071963 0.75 SCN9A (0.56) SCN9ASIGMAR1NAMPTGAALMNA
SCHEMBL1709232 0.74 SCN9A (1.00) SCN9ANAMPTGAAPOLBACHE
SCHEMBL10072406 0.73 SCN9A (0.57) SCN9ASIGMAR1NAMPTPOLBACHE
SCHEMBL1709247 0.72 SCN9A (0.64) SCN9ASIGMAR1NAMPTHTTMEN1
SCHEMBL1709234 0.72 SCN9A (0.60) SCN9ANAMPTKDM4EHTTACHE
SCHEMBL10071962 0.71 SCN9A (0.57) SCN9ANAMPTACHEBACE1
SCHEMBL1709212 0.70 ACHE (0.45) SCN9ASIGMAR1KDM4EGAALMNA
SCHEMBL4216674 0.68 ALDH1A1 (0.50) SIGMAR1KDM4EGAALMNAPOLB
SCHEMBL20641661 0.68 CHRM4 (0.73) SCN9AACHE

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012047703-A2 CYCLOPROPYL-SPIRO-PIPERIDINES USEFUL AS SODIUM CHANNEL BLOCKERS SCHERING CORPORATION (US) 2012-04-12 WO disclosed