SCHEMBL1709505

SCHEMBL1709505

O=C(O)C[C@H]1CCC[C@@H](N(CCC(F)(F)F)Cc2ccccc2)[C@@H]1c1ccc(C(F)(F)F)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HDAC4 P56524 1/20 0.40
DGAT1 O75907 1/20 0.35
HRH3 Q9Y5N1 1/20 0.34
SLC6A2 P23975 1/20 0.34
SLC6A4 P31645 1/20 0.34
PSEN1 P49768 2/20 0.34
PSEN2 P49810 2/20 0.34
APH1B Q8WW43 2/20 0.34
NCSTN Q92542 2/20 0.34
APH1A Q96BI3 2/20 0.34
PSENEN Q9NZ42 2/20 0.34
KCNH2 Q12809 1/20 0.33
TACR1 P25103 2/20 0.33
MEN1 O00255 1/20 0.32
ALDH1A1 P00352 1/20 0.32
KMT2A Q03164 1/20 0.32
TRPM8 Q7Z2W7 1/20 0.32
CHRM4 P08173 1/20 0.32
KDM1A O60341 1/20 0.32
MAOA P21397 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10033123 0.89 PSEN1 (0.41) HDAC4DGAT1HRH3PSEN1PSEN2
SCHEMBL10032999 0.74 SCN9A (0.43) CHRM4LIPE
SCHEMBL10033002 0.72 SLC6A2 (0.37) SLC6A2SLC6A4KCNH2TACR1ALDH1A1
SCHEMBL1709388 0.68 MAOA (0.45) HDAC4HRH3KCNH2TACR1KDM1A
SCHEMBL27403931 0.67 HRH3 (0.48) HDAC4DGAT1HRH3PSEN1PSEN2
SCHEMBL2316015 0.66 PSEN1 (0.43) DGAT1HRH3PSEN1PSEN2APH1B
SCHEMBL1709467 0.66 TACR1 (0.41) SLC6A2SLC6A4KCNH2TACR1MEN1
SCHEMBL10033174 0.65 CFTR (0.41) SLC6A4TACR1MEN1ALDH1A1KMT2A
SCHEMBL1709405 0.64 TACR1 (0.38) DGAT1PSEN1PSEN2APH1BNCSTN
SCHEMBL20516506 0.64 HCRTR1 (0.48)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012046771-A1 CYCLOALKANE COMPOUND アステラス製薬株式会社 (JP) 2012-04-12 WO disclosed