SCHEMBL1710177

SCHEMBL1710177

COc1cc(Cl)c(COC2CCCCO2)c(Cn2cccc(C#N)c2=O)n1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
P2RX3 P56373 7/20 0.34
ALDH1A1 P00352 2/20 0.33
KDM4E B2RXH2 1/20 0.33
GLA P06280 1/20 0.33
GAA P10253 1/20 0.33
HPGD P15428 1/20 0.33
NPC1 O15118 1/20 0.32
RAB9A P51151 1/20 0.32
CYP3A4 P08684 3/20 0.31
DPP4 P27487 3/20 0.31
KDM4C Q9H3R0 1/20 0.31
LMNA P02545 1/20 0.31
PDE4A P27815 2/20 0.31
PDE4B Q07343 2/20 0.31
PDE4C Q08493 2/20 0.31
PDE4D Q08499 2/20 0.31
CCNA2 P20248 1/20 0.30
CDK2 P24941 1/20 0.30
CCNA1 P78396 1/20 0.30
CDK5 Q00535 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1722176 0.97 P2RX3 (0.33) P2RX3ALDH1A1KDM4EGLAGAA
SCHEMBL1710193 0.83 CCNA2 (0.30) CCNA2CDK2CCNA1CDK5CDK5R1
SCHEMBL1710219 0.78 MBOAT4 (0.37) NPC1RAB9AKDM4CPDE4APDE4B
SCHEMBL1710353 0.77 NPC1 (0.39) P2RX3NPC1RAB9AKDM4CPDE4A
SCHEMBL1710329 0.74 KDM4E (0.32) ALDH1A1KDM4EGLAGAAHPGD
SCHEMBL1710200 0.73 NPC1 (0.41) P2RX3NPC1RAB9AKDM4CPDE4A
SCHEMBL1710191 0.69
SCHEMBL1710278 0.69 NPC1 (0.38) P2RX3NPC1RAB9AKDM4CPDE4A
SCHEMBL1722853 0.68 BDKRB2 (0.48) CYP3A4
SCHEMBL1710178 0.68 KDM4E (0.40) ALDH1A1KDM4EGAAHPGDNPBWR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344477-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS Jerini AG (DE) 2011-07-20 EP disclosed
WO-2010031589-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-03-25 WO disclosed