SCHEMBL1710219

SCHEMBL1710219

COc1cc(Cl)c(COC2CCCCO2)c(Cc2ccc(C#N)c(=O)[nH]2)n1

nearest known ligand 0.37

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
MBOAT4 Q96T53 1/20 0.37
IDH1 O75874 14/20 0.34
PDE4A P27815 1/20 0.33
PDE4B Q07343 1/20 0.33
PDE4C Q08493 1/20 0.33
PDE4D Q08499 1/20 0.33
NPC1 O15118 1/20 0.33
RAB9A P51151 1/20 0.33
XDH P47989 1/20 0.32
KDM4C Q9H3R0 1/20 0.31
CCNA2 P20248 1/20 0.31
CDK2 P24941 1/20 0.31
CCNA1 P78396 1/20 0.31
CDK5 Q00535 1/20 0.31
CDK5R1 Q15078 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1710225 0.90 MBOAT4 (0.40) MBOAT4IDH1NPC1RAB9AXDH
SCHEMBL1710449 0.80 MBOAT4 (0.40) MBOAT4IDH1XDH
SCHEMBL1710177 0.78 P2RX3 (0.34) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL1710353 0.77 NPC1 (0.39) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL1710191 0.76
SCHEMBL1722176 0.76 P2RX3 (0.33) NPC1RAB9A
SCHEMBL1710200 0.74 NPC1 (0.41) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL1710193 0.73 CCNA2 (0.30) CCNA2CDK2CCNA1CDK5CDK5R1
SCHEMBL1710278 0.70 NPC1 (0.38) PDE4APDE4BPDE4CPDE4DNPC1
SCHEMBL1710284 0.69 BDKRB2 (0.56) MBOAT4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344477-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS Jerini AG (DE) 2011-07-20 EP disclosed
WO-2010031589-A1 SMALL MOLECULE BRADYKININ B2 RECEPTOR MODULATORS JERINI AG (DE) 2010-03-25 WO disclosed