SCHEMBL17181769

SCHEMBL17181769

Nc1ccnc(B(O)O)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ASIC3 Q9UHC3 3/20 0.41
ALDH1A1 P00352 3/20 0.40
KDM4E B2RXH2 3/20 0.40
ENPP2 Q13822 1/20 0.40
MAPT P10636 2/20 0.35
TSHR P16473 2/20 0.35
SMN1; SMN2 Q16637 2/20 0.35
MEN1 O00255 2/20 0.35
KMT2A Q03164 2/20 0.35
CHRM1 P11229 2/20 0.35
LMNA P02545 1/20 0.35
CYP2D6 P10635 1/20 0.35
MAPK1 P28482 1/20 0.35
KCNA1 Q09470 1/20 0.35
PLG P00747 1/20 0.33
F12 P00748 1/20 0.33
F11 P03951 1/20 0.33
KLKB1 P03952 1/20 0.33
PRSS1 P07477 1/20 0.33
PRSS2 P07478 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL28507681 0.74 KDM4E (0.47) ALDH1A1KDM4ETSHRSMN1; SMN2MEN1
SCHEMBL28668509 0.74 ENPP2 (0.38) ALDH1A1KDM4EENPP2SMN1; SMN2MEN1
SCHEMBL1404632 0.74 ENPP2 (0.38) ALDH1A1KDM4EENPP2TSHRPLG
SCHEMBL29954387 0.73 KMO (0.34) ALDH1A1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL1843516 0.73 KMO (0.34) ALDH1A1SMN1; SMN2MEN1KMT2ALMNA
SCHEMBL29952078 0.73 UHRF1 (0.50) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL1843835 0.73 UHRF1 (0.50) ALDH1A1KDM4ESMN1; SMN2MEN1KMT2A
SCHEMBL4484450 0.73 NR4A2 (0.38) ALDH1A1ENPP2MAPTSMN1; SMN2LMNA
SCHEMBL2814691 0.70 NUDT1 (0.30) ASIC3
SCHEMBL29806893 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
CN-116178337-B Benzodiazepine compounds and their use as Rho kinase inhibitors 成都奥睿药业有限公司 2025-04-25 CN disclosed
EP-4527393-A1 SURFACE-MODIFIED NANODIAMOND Kyoto University (JP) 2025-03-26 EP disclosed
WO-2023223962-A1 SURFACE-MODIFIED NANODIAMOND 国立大学法人京都大学 2023-11-23 WO disclosed
WO-2023093787-A1 BENZODIAZEPINE COMPOUND AND APPLICATION THEREOF AS RHO KINASE INHIBITOR 成都奥睿药业有限公司 2023-06-01 WO disclosed
CN-116178337-A Benzodiazepine compounds and their use as Rho kinase inhibitors 成都奥睿药业有限公司 2023-05-30 CN disclosed
US-20220340893-A1 BI-FUNCTIONAL COMPLEXES AND METHODS FOR MAKING AND USING SUCH COMPLEXES NUEVOLUTION A/S (DK) 2022-10-27 US disclosed
EP-2925319-B1 MIXED LINEAGE KINASE INHIBITORS FOR HIV/AIDS THERAPIES UNIV ROCHESTER (US) 2019-01-09 EP disclosed
EP-3037421-A1 MLK INHIBITORS AND METHODS OF USE University Of Rochester (US) 2016-06-29 EP disclosed
EP-2379561-B1 MLK INHIBITORS AND METHODS OF USE UNIV ROCHESTER (US) 2015-11-04 EP disclosed
US-20150297587-A1 MIXED LINEAGE KINASE INHIBITORS FOR HIV/AIDS THERAPIES NATIONAL INSTITUTES OF HEALTH (NIH), U.S. DEPT. OF HEALTH AND HUMAN SERVICES (DHHS), U.S. GOVERNMENT 2015-10-22 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150297587-A1 MIXED LINEAGE KINASE INHIBITORS FOR HIV/AIDS THERAPIES MLKL, MARCKS, MAP3K4 ASIC3 4295/4885ALDH1A1 4296/4885KDM4E 2231/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.