SCHEMBL172150

SCHEMBL172150

CCc1nn2ccc3c(c2c1C(=O)O)CCO3

nearest known ligand 0.63

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 17/20 0.63
MTNR1A P48039 15/20 0.63
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
DRD3 P35462 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL127145 0.90 MTNR1B (0.66) MTNR1BMTNR1A
SCHEMBL128531 0.86 MTNR1A (0.59) MTNR1BMTNR1A
SCHEMBL172456 0.84 MTNR1B (0.60) MTNR1BMTNR1A
SCHEMBL127261 0.81 MTNR1B (0.67) MTNR1BMTNR1AHTR2A
SCHEMBL126819 0.78 MTNR1B (0.59) MTNR1BMTNR1AHTR2A
SCHEMBL172399 0.78 MTNR1A (0.67) MTNR1BMTNR1ADRD2HTR2ADRD3
SCHEMBL172381 0.78 MTNR1B (0.62) MTNR1BMTNR1A
SCHEMBL123197 0.78 MTNR1A (1.00) MTNR1BMTNR1A
SCHEMBL124885 0.77 MTNR1B (1.00) MTNR1BMTNR1A
SCHEMBL124731 0.77 MTNR1A (0.67) MTNR1BMTNR1AHTR2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2100895-B1 TRICYCLIC COMPOUND AND MEDICAL USE THEREOF TAKEDA PHARMACEUTICAL (JP) 2012-03-07 EP disclosed