SCHEMBL1723018

SCHEMBL1723018

COCC(=O)C1=C(OC(C)=O)N(C)N(c2ccc(F)cc2Cl)C1O

nearest known ligand 0.35

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 1/20 0.35
GRM5 P41594 2/20 0.33
P2RX7 Q99572 7/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1723076 0.71 GRM5 (0.37) NPSR1GRM5P2RX7
SCHEMBL2845682 0.69 GRM5 (0.34) NPSR1GRM5P2RX7
SCHEMBL2849167 0.65 GRM5 (0.35) GRM5P2RX7
SCHEMBL1723074 0.62 P2RX7 (0.36) GRM5P2RX7
SCHEMBL3728350 0.61 KDM4E (0.44)
SCHEMBL3250915 0.61 MARS1 (0.39) GRM5P2RX7
SCHEMBL1722408 0.59 MARS1 (0.37) P2RX7
SCHEMBL3328392 0.58 CYP4F2 (0.44)
SCHEMBL31711605 0.57 CES2 (0.55)
SCHEMBL2031215 0.56 SMN1; SMN2 (0.45)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344492-A1 PYRAZOLO PYRIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GenKyoTex SA (CH) 2011-07-20 EP disclosed
WO-2010035221-A1 PYRAZOLO PYRIDINE DERIVATIVES AS NADPH OXIDASE INHIBITORS GENKYOTEX SA (CH) 2010-04-01 WO disclosed