SCHEMBL17232186

SCHEMBL17232186

c1ccc(-c2nc(-c3ccccc3)nc(-c3cccc(-c4cccc5c4oc4ccccc45)c3)n2)cc1

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALOX5 P09917 2/20 0.57
GGPS1 O95749 1/20 0.48
PTGES2 Q9H7Z7 1/20 0.45
MAPT P10636 7/20 0.42
PRKDC P78527 4/20 0.42
ALDH1A1 P00352 4/20 0.41
TSHR P16473 3/20 0.41
HPGD P15428 2/20 0.41
KDM4E B2RXH2 2/20 0.41
POLB P06746 2/20 0.41
PIK3CD O00329 1/20 0.41
PIK3CB P42338 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
HSD17B10 Q99714 2/20 0.40
LMNA P02545 2/20 0.40
KMT2A Q03164 2/20 0.40
TP53 P04637 1/20 0.40
NFKB1 P19838 1/20 0.40
MAPK1 P28482 1/20 0.40
NFKB2 Q00653 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL21563826 1.00 ALOX5 (0.57) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL21168062 1.00 ALOX5 (0.57) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL21563827 0.99 ALOX5 (0.59) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL19196619 0.99 ALOX5 (0.56) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL23008289 0.97 ALOX5 (0.58) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL16573901 0.97 ALOX5 (0.55) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL21563737 0.97 ALOX5 (0.55) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL15501889 0.97 ALOX5 (0.55) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL18216730 0.97 ALOX5 (0.55) ALOX5GGPS1PTGES2MAPTPRKDC
SCHEMBL21707165 0.97 ALOX5 (0.58) ALOX5GGPS1PTGES2MAPTPRKDC

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 18 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3533794-B1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2022-02-23 EP disclosed
US-20210340103-A1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT USING SAME, AND ELECTRONIC APPARATUS THEREOF DUK SAN NEOLUX CO., LTD (KR) 2021-11-04 US disclosed
US-20210184129-A1 COMPOUND FOR ORGANIC ELECTRONIC ELEMENT, ORGANIC ELECTRONIC ELEMENT USING SAME AND ELECTRONIC DEVICE THEREOF DUK SAN NEOLUX CO., LTD (KR) 2021-06-17 US disclosed
US-10985330-B2 Materials for electronic devices MERCK PATENT GMBH (DE) 2021-04-20 US disclosed
US-20210028370-A1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT USING THE SAME, AND ELECTRONIC DEVICE THEREFOR DUK SAN NEOLUX CO., LTD. (KR) 2021-01-28 US disclosed
WO-2019190101-A1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT USING SAME, AND ELECTRONIC DEVICE THEREFOR 덕산네오룩스 주식회사 2019-10-03 WO disclosed
EP-3533794-A2 MATERIALS FOR ELECTRONIC DEVICES Merck Patent GmbH (DE) 2019-09-04 EP disclosed
US-10355223-B2 Materials for electronic devices MERCK PATENT GMBH (DE) 2019-07-16 US disclosed
EP-3137458-B1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2019-04-24 EP disclosed
US-20170244044-A1 ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2017-08-24 US disclosed
US-20170244044-A1 ORGANIC ELECTROLUMINESCENT ELEMENT AND ELECTRONIC DEVICE IDEMITSU KOSAN CO., LTD. (JP) 2017-08-24 US disclosed
US-20170222160-A1 ORGANIC LIGHT EMITTING COMPOUNDS AND ORGANIC LIGHT EMITTING DEVICES INCLUDING THE SAME SFC CO., LTD. (KR) 2017-08-03 US disclosed
US-20170222160-A1 ORGANIC LIGHT EMITTING COMPOUNDS AND ORGANIC LIGHT EMITTING DEVICES INCLUDING THE SAME SFC CO., LTD. (KR) 2017-08-03 US disclosed
US-20170062736-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2017-03-02 US disclosed
US-20170062736-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2017-03-02 US disclosed
US-20160329506-A1 ORGANIC COMPOUND, ORGANIC OPTOELECTRONIC DEVICE, AND DISPLAY DEVICE SAMSUNG SDI CO., LTD. (KR) 2016-11-10 US disclosed
US-20160329506-A1 ORGANIC COMPOUND, ORGANIC OPTOELECTRONIC DEVICE, AND DISPLAY DEVICE SAMSUNG SDI CO., LTD. (KR) 2016-11-10 US disclosed
WO-2015165563-A1 MATERIALS FOR ELECTRONIC DEVICES MERCK PATENT GMBH (DE) 2015-11-05 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (8 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160329506-A1 ORGANIC COMPOUND, ORGANIC OPTOELECTRONIC DEVICE, AND DISPLAY DEVICE OCIAD1, OXER1, OR10J3 ALOX5 525/4885GGPS1 801/4885PTGES2 2438/4885
US-20170222160-A1 ORGANIC LIGHT EMITTING COMPOUNDS AND ORGANIC LIGHT EMITTING DEVICES INCLUDING THE SAME ALDH1A2, LAGE3, AOX1 ALOX5 446/4885GGPS1 515/4885PTGES2 953/4885
US-20170062736-A1 MATERIALS FOR ELECTRONIC DEVICES EPHA3, EPHA6, DDT ALOX5 3691/4885GGPS1 2010/4885PTGES2 1987/4885
US-20210028370-A1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT USING THE SAME, AND ELECTRONIC DEVICE THEREFOR OR51E2, WEE1, SLC39A11 ALOX5 936/4885GGPS1 824/4885PTGES2 2276/4885
US-20210340103-A1 COMPOUND FOR ORGANIC ELECTRIC ELEMENT, ORGANIC ELECTRIC ELEMENT USING SAME, AND ELECTRONIC APPARATUS THEREOF OR51E2, SLC39A11, WEE1 ALOX5 969/4885GGPS1 831/4885PTGES2 1450/4885
US-10355223-B2 Materials for electronic devices EPHA3, EPHA6, DDT ALOX5 3691/4885GGPS1 2010/4885PTGES2 1987/4885
US-20210184129-A1 COMPOUND FOR ORGANIC ELECTRONIC ELEMENT, ORGANIC ELECTRONIC ELEMENT USING SAME AND ELECTRONIC DEVICE THEREOF OR51E2, SLC39A11, WEE1 ALOX5 784/4885GGPS1 782/4885PTGES2 1863/4885
US-10985330-B2 Materials for electronic devices EPHA3, EPHA6, DDT ALOX5 3691/4885GGPS1 2010/4885PTGES2 1987/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.