SCHEMBL1724178

SCHEMBL1724178

O=C(O)NCCC(O)c1cccc(SCC2CCC(F)(F)CC2)c1

nearest known ligand 0.46

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 3/20 0.35
AGTR2 P50052 1/20 0.34
ROCK1 Q13464 1/20 0.34
CCR5 P51681 4/20 0.33
P2RX7 Q99572 4/20 0.33
ATM Q13315 1/20 0.32
L3MBTL1 Q9Y468 1/20 0.32
KCNQ3 O43525 1/20 0.32
KCNQ2 O43526 1/20 0.32
KCNQ4 P56696 1/20 0.32
KCNQ5 Q9NR82 1/20 0.32
CTSK P43235 1/20 0.32
MAP1LC3B Q9GZQ8 1/20 0.31
MAP1LC3A Q9H492 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1710752 0.87 BCHE (0.38) AGTR2CTSK
SCHEMBL1724792 0.86 IL1B (0.36) ROCK2P2RX7
SCHEMBL16031201 0.85 GCK (0.36) ROCK2AGTR2L3MBTL1MAP1LC3BMAP1LC3A
SCHEMBL16031904 0.85 AGTR2 (0.35) AGTR2CTSKMAP1LC3BMAP1LC3A
SCHEMBL1710613 0.85 PNMT (0.32) ROCK2AGTR2
SCHEMBL16031844 0.80 HPGD (0.34) AGTR2CTSKMAP1LC3BMAP1LC3A
SCHEMBL3390167 0.78 CTSK (0.37) AGTR2CTSK
SCHEMBL13400259 0.78 HDAC6 (0.38) CTSK
SCHEMBL13400239 0.78 HDAC6 (0.38) CTSK
SCHEMBL1710885 0.77 BCHE (0.37) CTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2344451-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS Acucela, Inc. (US) 2011-07-20 EP disclosed
WO-2010028088-A2 SULFUR-LINKED COMPOUNDS FOR TREATING OPTHALMIC DISEASES AND DISORDERS ACUCELA, INC. (US) 2010-03-11 WO disclosed