Propomocarb

Propomocarb

SCHEMBL1724451

CC(=O)O.CCCOC(=O)NCCCN(C)C

nearest known ligand 0.56

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA2AADRA2BADRA2CADRB2AGTR1AVPR1AAVPR1BAVPR2BDKRB2CALCRCHRNA3CHRNB4ESR1ESR2GHSRGNRHRGSC1HSPA8MALT1MC1RMC4RNOS1NOS2NOS3OPRK1OXTRRAMP1RAMP2RAMP3SCN5ASSTR1SSTR2SSTR3SSTR4SSTR5dacAdacBdacCfolPftsImrcAmrcBmrdArplArplBrplCrplDrplErplFrplJrplKrplLrplMrplNrplOrplPrplQrplRrplSrplTrplUrplVrplWrplXrplYrpmArpmBrpmCrpmDrpmErpmFrpmGrpmHrpmIrpmJrpsArpsBrpsCrpsDrpsErpsFrpsGrpsHrpsIrpsJrpsKrpsLrpsMrpsNrpsOrpsPrpsQrpsRrpsSrpsTrpsUykgMykgO

The experimentally established mechanism targets of Propomocarb. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
CHRNB4 known ✓ P30926 1/20 0.45
CHRNA3 known ✓ P32297 1/20 0.45
ACHE P22303 14/20 0.56
DNM1 Q05193 1/20 0.47
CHRNB2 P17787 1/20 0.45
CHRNA4 P43681 1/20 0.45
TLR2 O60603 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Propomocarb SCHEMBL21077 0.95 ACHE (0.61) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL11597864 0.94 ACHE (0.56) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL17095085 0.93 ACHE (0.59) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL68988 0.93 ACHE (0.59) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL8437517 0.93 ACHE (0.59) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL11598946 0.92 ACHE (0.54) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL28227333 0.92 ACHE (0.62) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL11599265 0.91 ACHE (0.53) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL6552410 0.90 ACHE (0.56) ACHEDNM1CHRNB2CHRNB4CHRNA3
Propomocarb SCHEMBL6552413 0.90 ACHE (0.56) ACHEDNM1CHRNB2CHRNB4CHRNA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2540716-B1 TETRAZOLYLOXIME DERIVATIVE OR A SALT THEREOF, AND GERMICIDE NIPPON SODA CO (JP) 2015-11-11 EP disclosed
US-9156816-B2 Tetrazolyloxime derivative or salt thereof and fungicide NIPPON SODA CO., LTD. (JP) 2015-10-13 US disclosed
EP-2177519-B1 TETRAZOYLOXIME DERIVATIVE AND PLANT DISEASE CONTROL AGENT NIPPON SODA CO (JP) 2015-05-27 EP disclosed
US-9029552-B2 Tetrazoyloxime derivative and plant disease control agent NIPPON SODA CO., LTD. (JP) 2015-05-12 US disclosed
US-8710084-B2 Tetrazolyl oxime derivative, salt thereof, and plant disease control agent NIPPON SODA CO., LTD. (JP) 2014-04-29 US disclosed
US-20140005385-A1 TETRAZOYLOXIME DERIVATIVE AND PLANT DISEASE CONTROL AGENT NIPPON SODA CO., LTD. (JP) 2014-01-02 US disclosed
EP-2669282-A1 Tetrazoyloxime derivative and plant disease control agent NIPPON SODA CO., LTD. (JP) 2013-12-04 EP disclosed
EP-2404917-B1 TETRAZOLYL OXIME DERIVATIVE, SALT THEREOF, AND PLANT DISEASE CONTROL AGENT NIPPON SODA CO (JP) 2013-09-04 EP disclosed
EP-2540716-A1 TETRAZOLYLOXIME DERIVATIVE OR A SALT THEREOF, AND GERMICIDE Nippon Soda Co., Ltd. (JP) 2013-01-02 EP disclosed
US-20120309972-A1 TETRAZOLYLOXIME DERIVATIVE OR SALT THEREOF AND FUNGICIDE NIPPON SODA CO., LTD. (JP) 2012-12-06 US disclosed
EP-2404917-A1 TETRAZOYL OXIME DERIVATIVE, SALT THEREOF, AND PLANT DISEASE CONTROL AGENT Nippon Soda Co., Ltd. (JP) 2012-01-11 EP disclosed
US-20110313152-A1 TETRAZOLYL OXIME DERIVATIVE, SALT THEREOF, AND PLANT DISEASE NIPPON SODA CO., LTD. (JP) 2011-12-22 US disclosed
US-20100137594-A1 TETRAZOYLOXIME DERIVATIVE AND PLANT DISEASE CONTROL AGENT NIPPON SODA CO., LTD. (JP) 2010-06-03 US disclosed
EP-2177519-A1 TETRAZOYLOXIME DERIVATIVE AND PLANT DISEASE CONTROL AGENT Nippon Soda Co., Ltd. (JP) 2010-04-21 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20120309972-A1 TETRAZOLYLOXIME DERIVATIVE OR SALT THEREOF AND FUNGICIDE AS3MT, PRXL2A, TH CHRNB4 4527/4885CHRNA3 4394/4885ACHE 3666/4885
US-20110313152-A1 TETRAZOLYL OXIME DERIVATIVE, SALT THEREOF, AND PLANT DISEASE H1-10, H1-0, OXSR1 CHRNB4 3700/4885CHRNA3 2445/4885ACHE 3106/4885
US-20140005385-A1 TETRAZOYLOXIME DERIVATIVE AND PLANT DISEASE CONTROL AGENT PAOX, BROX, TTI2 CHRNB4 4779/4885CHRNA3 4742/4885ACHE 1398/4885
US-20100137594-A1 TETRAZOYLOXIME DERIVATIVE AND PLANT DISEASE CONTROL AGENT PAOX, H1-10, HAX1 CHRNB4 3937/4885CHRNA3 3512/4885ACHE 2082/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.