SCHEMBL17284643

SCHEMBL17284643

NC1CCN(CCCN2CCN(Cc3ccccc3)C2=O)CC1

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
DRD3 P35462 4/20 0.54
KCNH2 Q12809 4/20 0.54
POLB P06746 1/20 0.49
CYP2D6 P10635 1/20 0.49
CYP2C9 P11712 1/20 0.49
CYP2C19 P33261 1/20 0.49
KMT2A Q03164 1/20 0.49
DRD2 P14416 1/20 0.44
MAPK1 P28482 1/20 0.43
SIGMAR1 Q99720 1/20 0.42
CCR3 P51677 1/20 0.41
PARP1 P09874 1/20 0.41
PARP2 Q9UGN5 1/20 0.41
SLC6A2 P23975 1/20 0.41
SLC6A4 P31645 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17285906 0.87 ACHE (0.57) DRD3KCNH2POLBCYP2D6CYP2C9
SCHEMBL22878313 0.87 DRD3 (0.54) DRD3KCNH2POLBCYP2D6CYP2C9
SCHEMBL18876620 0.85 KCNH2 (0.52) DRD3KCNH2POLBCYP2D6CYP2C9
SCHEMBL17281928 0.84 DRD3 (0.51) DRD3KCNH2POLBCYP2D6CYP2C9
SCHEMBL4873038 0.79 DRD3 (0.60) DRD3KCNH2POLBCYP2D6CYP2C9
SCHEMBL29450073 0.76 KMT2A (0.76) DRD3KCNH2POLBCYP2D6CYP2C9
SCHEMBL16416392 0.76 KMT2A (0.76) DRD3KCNH2POLBCYP2D6CYP2C9
SCHEMBL17284644 0.76 GNAI3 (0.47) DRD3KCNH2KMT2ADRD2MAPK1
SCHEMBL1587336 0.75 SIGMAR1 (0.70) KCNH2POLBCYP2D6CYP2C19KMT2A
SCHEMBL42207 0.75 ACHE (0.67) DRD3DRD2SIGMAR1CCR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2015177326-A1 5-CHLORO-2-DIFLUOROMETHOXYPHENYL PYRAZOLOPYRIMIDINE COMPOUNDS WHICH ARE JAK INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2015-11-26 WO disclosed