SCHEMBL1728748

SCHEMBL1728748

CN(CCOc1ccc(-n2ccn(-c3ccc(Oc4ccccc4)cc3)c2=O)cc1)Cc1ccccc1

nearest known ligand 0.66

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
MCHR1 Q99705 4/20 0.66
KCNH2 Q12809 3/20 0.66
TSHR P16473 1/20 0.57
LTA4H P09960 1/20 0.50
KDM4E B2RXH2 1/20 0.48
ALDH1A1 P00352 1/20 0.48
ATM Q13315 1/20 0.48
BCHE P06276 1/20 0.47
ACHE P22303 1/20 0.47
MAOB P27338 1/20 0.47
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1728610 0.90 KCNH2 (0.57) MCHR1KCNH2TSHRLTA4HACHE
SCHEMBL1728135 0.87 LTA4H (0.51) MCHR1KCNH2TSHRLTA4H
SCHEMBL6081348 0.87 LTA4H (0.51) MCHR1KCNH2TSHRLTA4H
SCHEMBL1728669 0.87 LTA4H (0.68) MCHR1KCNH2LTA4HKDM4EALDH1A1
SCHEMBL1728580 0.85 LTA4H (0.51) MCHR1KCNH2LTA4HALDH1A1MEN1
SCHEMBL1729935 0.81 MCHR1 (0.45) MCHR1KCNH2LTA4HMEN1KMT2A
SCHEMBL1728641 0.81 GNRHR (0.48) MCHR1KCNH2TSHRLTA4HKDM4E
SCHEMBL1728493 0.80 MCHR1 (0.78) MCHR1KCNH2LTA4H
SCHEMBL1728658 0.80 LTA4H (0.70) MCHR1KCNH2LTA4H
SCHEMBL2893078 0.80 MCHR1 (1.00) MCHR1KCNH2TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1551810-B1 DIARYL-SUBSTITUTED CYCLIC UREA DERIVATIVES HAVING AN MCH-MODULATORY EFFECT SANOFI AVENTIS DEUTSCHLAND (DE) 2011-11-30 EP disclosed
US-7141561-B2 Substituted diaryl heterocycles, process for their preparation and their use as medicaments SANOFI-AVENTIS DEUTSCHLAND GMBH (DE) 2006-11-28 US disclosed