SCHEMBL17329014

SCHEMBL17329014

Cc1cc2c(Cl)nccc2o1

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP1A1 P04798 5/20 0.41
CYP1A2 P05177 5/20 0.41
CYP1B1 Q16678 5/20 0.41
F2RL3 Q96RI0 3/20 0.41
POLB P06746 1/20 0.35
L3MBTL1 Q9Y468 1/20 0.35
LMNA P02545 2/20 0.35
ALDH1A1 P00352 1/20 0.35
KMT2A Q03164 1/20 0.35
GPR55 Q9Y2T6 1/20 0.35
CYP3A4 P08684 1/20 0.34
MAPT P10636 1/20 0.34
APEX1 P27695 1/20 0.34
MAPK1 P28482 1/20 0.34
PMP22 Q01453 1/20 0.34
NPC1 O15118 1/20 0.34
RAB9A P51151 1/20 0.34
RXFP1 Q9HBX9 1/20 0.34
HTR2A P28223 1/20 0.33
HTR2C P28335 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30110720 1.00 CYP1A1 (0.41) CYP1A1CYP1A2CYP1B1F2RL3POLB
SCHEMBL17531152 0.80 POLB (0.43) CYP1A1CYP1A2CYP1B1POLBL3MBTL1
SCHEMBL31393644 0.78 F2RL3 (0.42) CYP1A2F2RL3POLBL3MBTL1LMNA
SCHEMBL21076531 0.78 F2RL3 (0.39) F2RL3POLBL3MBTL1LMNAALDH1A1
SCHEMBL8269242 0.77 MET (0.44) CYP1A1CYP1A2CYP1B1KMT2AHTR2A
SCHEMBL29210400 0.77 F2RL3 (0.47) F2RL3POLBL3MBTL1LMNAALDH1A1
SCHEMBL21076479 0.77 F2RL3 (0.39) F2RL3HTR2AHTR2C
SCHEMBL22490021 0.74 HTR2A (0.37) CYP1A1CYP1A2CYP1B1ALDH1A1NPC1
SCHEMBL18678557 0.74 CYP2A6 (0.42) F2RL3POLBL3MBTL1LMNAALDH1A1
SCHEMBL15349692 0.74 ALDH1A1 (0.51) F2RL3POLBL3MBTL1LMNAALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 13 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-12522595-B2 Bicyclic ether O-glycoprotein-2-acetamido-2-deoxy-3-D-glucopyranosidase inhibitors BIOGEN MA INC. (US) 2026-01-13 US disclosed
EP-4169575-B1 CONDENSED RING COMPOUNDS THAT INHIBIT H-PGDS SATO PHARMA (JP) 2026-01-07 EP disclosed
US-20230339937-A1 CONDENSED RING COMPOUNDS THAT INHIBIT H-PGDS SATO PHARMACEUTICAL CO., LTD. (JP) 2023-10-26 US disclosed
EP-4169575-A1 CONDENSED RING COMPOUNDS THAT INHIBIT H-PGDS Sato Pharmaceutical Co., Ltd. (JP) 2023-04-26 EP disclosed
CN-115667259-A Condensed ring compounds for inhibiting H-PGDS 佐藤制药株式会社 2023-01-31 CN disclosed
US-20220106305-A1 BICYCLIC ETHER O-GLYCOPROTEIN-2-ACETAMIDO-2-DEOXY-3-D-GLUCOPYRANOSIDASE INHIBITORS BIOGEN MA INC. 2022-04-07 US disclosed
EP-3921316-A1 BICYCLIC ETHER O-GLYCOPROTEIN-2-ACETAMIDO-2-DEOXY-3-D-GLUCOPYRANOSIDASE INHIBITORS Biogen MA Inc. (US) 2021-12-15 EP disclosed
EP-2955185-B1 POLYCYCLIC SUBSTITUTED PYRAZOLE KINASE ACTIVITY INHIBITORS AND USE THEREOF SHANGHAI FOSUN PHARMACEUTICAL DEV CO LTD (CN) 2021-01-06 EP disclosed
WO-2020163193-A1 BICYCLIC ETHER O-GLYCOPROTEIN-2-ACETAMIDO-2-DEOXY-3-D-GLUCOPYRANOSIDASE INHIBITORS BIOGEN MA INC. (US) 2020-08-13 WO disclosed
WO-2018029288-A1 SULFONYL PYRIDYL TRP INHIBITORS F. HOFFMANN-LA ROCHE AG (CH) 2018-02-15 WO disclosed
US-9550792-B2 Polycyclic substituted pyrazole kinase activity inhibitors and use thereof SHANGHAI FOSUN PHARMACEUTICAL DEVELOPMENT CO., LTD. (CN) 2017-01-24 US disclosed
US-20150368259-A1 Polycyclic Substituted Pyrazole Kinase Activity Inhibitors and Use Thereof SHANGHAI FOSUN PHARMACEUTICAL DEVELOPMENT CO., LTD. (CN) 2015-12-24 US disclosed
EP-2955185-A1 POLYCYCLIC SUBSTITUTED PYRAZOLE KINASE ACTIVITY INHIBITORS AND USE THEREOF China Pharmaceutical University (CN) 2015-12-16 EP disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20150368259-A1 Polycyclic Substituted Pyrazole Kinase Activity Inhibitors and Use Thereof MAP3K5, MAP3K19, MAP3K3 CYP1A1 2515/4885CYP1A2 1733/4885CYP1B1 1840/4885
US-20220106305-A1 BICYCLIC ETHER O-GLYCOPROTEIN-2-ACETAMIDO-2-DEOXY-3-D-GLUCOPYRANOSIDASE INHIBITORS ENGASE, UGGT1, MGAT3 CYP1A1 250/4885CYP1A2 160/4885CYP1B1 393/4885
US-20230339937-A1 CONDENSED RING COMPOUNDS THAT INHIBIT H-PGDS HPGDS, PTGS1, PTGIS CYP1A1 327/4885CYP1A2 438/4885CYP1B1 498/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.