SCHEMBL1734498

SCHEMBL1734498

CCC(CC1CC1)Nc1nc(C(N)=O)cc(-c2ccccc2OC)n1

nearest known ligand 0.47

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
VCP P55072 2/20 0.47
LRRK2 Q5S007 2/20 0.41
ADORA1 P30542 4/20 0.41
ADORA3 P0DMS8 4/20 0.41
ADORA2A P29274 2/20 0.40
CCNT1 O60563 1/20 0.39
CDK9 P50750 1/20 0.39
AGER Q15109 1/20 0.39
ALDH1A1 P00352 1/20 0.38
HPGD P15428 1/20 0.38
FPR2 P25090 1/20 0.38
SCN9A Q15858 1/20 0.38
ABL1 P00519 4/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734296 0.84 KDM4E (0.48) VCPADORA1ADORA3ADORA2AALDH1A1
SCHEMBL1735526 0.83 SCN9A (0.49) VCPADORA3ALDH1A1HPGDFPR2
SCHEMBL1733485 0.82 VCP (0.49) VCPLRRK2ADORA1ADORA3ADORA2A
SCHEMBL1734652 0.73 VCP (0.46) VCPADORA1ADORA3ADORA2ACCNT1
SCHEMBL1734302 0.73 MEN1 (0.51) VCPALDH1A1HPGD
SCHEMBL1735530 0.73 ADORA1 (0.46) VCPADORA1ADORA3ADORA2A
SCHEMBL1735520 0.73 KDM4E (0.56) ADORA1ADORA3ADORA2AALDH1A1HPGD
SCHEMBL1734497 0.72 KDM4E (0.47) VCPADORA1ADORA3ADORA2A
SCHEMBL2816888 0.71 HSP90AA1 (0.52) ADORA1ADORA3ADORA2ACCNT1CDK9
SCHEMBL1734511 0.70 KDM4E (0.66) ADORA1ADORA3ADORA2ACCNT1CDK9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed