SCHEMBL1735526

SCHEMBL1735526

CCC(CC1CC1)Nc1nc(C(N)=O)cc(-c2ccc(OC)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SCN9A Q15858 5/20 0.49
FPR2 P25090 1/20 0.49
ALDH1A1 P00352 3/20 0.48
HPGD P15428 2/20 0.48
KDM4E B2RXH2 1/20 0.48
TP53 P04637 1/20 0.48
GAA P10253 1/20 0.48
VCP P55072 4/20 0.46
ADORA3 P0DMS8 4/20 0.41
ADORA2B P29275 1/20 0.39
LMNA P02545 1/20 0.39
MAPT P10636 1/20 0.39
GSK3B P49841 1/20 0.39
EGFR P00533 1/20 0.38
KDR P35968 1/20 0.38
GLA P06280 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
GRM2 Q14416 1/20 0.38
PTGDR Q13258 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1733485 0.90 VCP (0.49) SCN9AFPR2KDM4ETP53VCP
SCHEMBL1734296 0.88 KDM4E (0.48) SCN9AFPR2ALDH1A1HPGDKDM4E
SCHEMBL1734498 0.83 VCP (0.47) SCN9AFPR2ALDH1A1HPGDVCP
SCHEMBL1734499 0.81 VCP (0.67) SCN9AALDH1A1HPGDKDM4ETP53
SCHEMBL1734297 0.78 TP53 (0.55) SCN9AFPR2ALDH1A1HPGDKDM4E
SCHEMBL1735520 0.76 KDM4E (0.56) SCN9AFPR2ALDH1A1HPGDKDM4E
SCHEMBL1735530 0.76 ADORA1 (0.46) VCPADORA3ADORA2B
SCHEMBL1734431 0.72 KDM4E (0.51) SCN9AFPR2ALDH1A1HPGDKDM4E
SCHEMBL1733597 0.72 TP53 (0.51) SCN9AFPR2ALDH1A1HPGDKDM4E
SCHEMBL1734563 0.71 KDM4E (0.51) ALDH1A1HPGDKDM4ETP53GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed