SCHEMBL1735530

SCHEMBL1735530

CCC(CC1CC1)Nc1nc(C(=O)N(C)C)cc(-c2ccccc2)n1

nearest known ligand 0.46

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ADORA1 P30542 9/20 0.46
VCP P55072 11/20 0.43
ADORA2A P29274 4/20 0.40
ADORA3 P0DMS8 3/20 0.40
ADORA2B P29275 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1734296 0.88 KDM4E (0.48) ADORA1VCPADORA2AADORA3ADORA2B
SCHEMBL1735526 0.76 SCN9A (0.49) VCPADORA3ADORA2B
SCHEMBL1733485 0.76 VCP (0.49) ADORA1VCPADORA2AADORA3ADORA2B
SCHEMBL1735520 0.76 KDM4E (0.56) ADORA1ADORA2AADORA3ADORA2B
SCHEMBL1734498 0.73 VCP (0.47) ADORA1VCPADORA2AADORA3
SCHEMBL1734431 0.71 KDM4E (0.51) ADORA1ADORA2AADORA3ADORA2B
SCHEMBL1734460 0.71 KDM4E (0.51) VCP
SCHEMBL1734181 0.70 KDM4E (0.50) ADORA1ADORA2AADORA3ADORA2B
SCHEMBL1734442 0.68 ALDH1A1 (0.49) VCP
SCHEMBL1734520 0.68 KDM4E (0.74) ADORA1ADORA2AADORA3ADORA2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1891018-B1 MODULATORS OF ATP-BINDING CASSETTE TRANSPORTERS VERTEX PHARMA (US) 2011-11-16 EP claimed
WO-2011131686-A1 A THERMALLY CONTROLLED ASSEMBLY NAPATECH A/S (DK) 2011-10-27 WO claimed