SCHEMBL17360345

SCHEMBL17360345

COCc1cc2c(ccn2C(=O)O)cc1OCc1ccccc1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SRD5A2 P31213 3/20 0.46
SRD5A1 P18405 2/20 0.46
BRD4 O60885 1/20 0.40
FFAR4 Q5NUL3 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.39
HPGD P15428 2/20 0.39
NPC1 O15118 1/20 0.39
RAB9A P51151 1/20 0.39
SMPD1 P17405 1/20 0.39
HDAC1 Q13547 1/20 0.39
HDAC8 Q9BY41 1/20 0.39
HDAC6 Q9UBN7 1/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
RXRA P19793 1/20 0.38
STAT3 P40763 1/20 0.38
HTT P42858 1/20 0.38
ELANE P08246 1/20 0.38
CTSG P08311 1/20 0.38
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17360243 0.88 ELANE (0.47) SRD5A2SRD5A1BRD4FFAR4SMN1; SMN2
SCHEMBL17360612 0.87 SRD5A1 (0.41) SRD5A2SRD5A1BRD4SMN1; SMN2HPGD
SCHEMBL15984664 0.77 ELANE (0.42) SRD5A2SRD5A1BRD4ELANECTSG
SCHEMBL29264495 0.75 SRD5A1 (0.49) SRD5A2SRD5A1BRD4SMN1; SMN2NPC1
SCHEMBL21274686 0.75 ALOX5 (0.54) SRD5A2HPGDNPC1RAB9AHDAC1
SCHEMBL5483649 0.75 SRD5A2 (0.57) SRD5A2HPGDNPC1RAB9AHDAC1
SCHEMBL18474166 0.73 SRD5A1 (0.55) SRD5A2SRD5A1SMN1; SMN2HPGDNPC1
SCHEMBL3916932 0.73 TUBB1 (0.58) SRD5A2SRD5A1SMN1; SMN2HPGDNPC1
SCHEMBL7163724 0.72 SRD5A1 (0.51) SRD5A2SRD5A1BRD4SMN1; SMN2HPGD
SCHEMBL3912610 0.70 TRPV3 (0.41) SRD5A2SRD5A1BRD4NPC1MRGPRX4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2960238-B1 MONOCYCLIC PYRIDINE DERIVATIVE EISAI R&D MAN CO LTD (JP) 2017-04-05 EP disclosed
EP-2960238-A1 MONOCYCLIC PYRIDINE DERIVATIVE Eisai R&D Management Co., Ltd. (JP) 2015-12-30 EP disclosed