SCHEMBL17400358

SCHEMBL17400358

CC1=CC=C(N2CCN(Cc3cc4[nH]c(=O)c5cc(F)ccc5n4c3)CC2)CC1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TNKS O95271 2/20 0.39
PARP1 P09874 10/20 0.37
KCNH2 Q12809 2/20 0.35
TNK1 Q13470 4/20 0.34
TNK2 Q07912 2/20 0.34
PARP2 Q9UGN5 2/20 0.33
TRPC5 Q9UL62 1/20 0.33
HTR6 P50406 1/20 0.33
DRD2 P14416 1/20 0.32
DRD4 P21917 1/20 0.32
DRD3 P35462 1/20 0.32
HTR3E A5X5Y0 1/20 0.32
HTR3B O95264 1/20 0.32
HTR1A P08908 1/20 0.32
HTR3A P46098 1/20 0.32
HTR3D Q70Z44 1/20 0.32
HTR3C Q8WXA8 1/20 0.32
HDAC1 Q13547 1/20 0.32
HDAC8 Q9BY41 1/20 0.32
HDAC6 Q9UBN7 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14647192 0.83 PARP1 (0.46) TNKSPARP1TNK1TNK2PARP2
SCHEMBL14647191 0.77 DRD4 (0.51) TNKSPARP1TNK1PARP2DRD2
SCHEMBL15979574 0.76 PARP1 (0.49) TNKSPARP1KCNH2TNK1TNK2
SCHEMBL14647183 0.74 PARP1 (0.46) PARP1TNK1TNK2DRD2DRD4
SCHEMBL14647166 0.74 PARP1 (0.49) PARP1KCNH2TNK1TNK2PARP2
SCHEMBL14647226 0.73 TNKS (0.43) TNKSPARP1HTR3EHTR3BHTR1A
SCHEMBL14647187 0.72 DRD4 (0.43) PARP1HTR6DRD2DRD4DRD3
SCHEMBL14647213 0.72 MAPK1 (0.49) PARP1HTR6DRD2DRD4DRD3
SCHEMBL14647239 0.70 KDM4E (0.46) DRD2DRD4DRD3HTR1A
SCHEMBL15979572 0.70 DRD2 (0.47) TNKSPARP1DRD2DRD4HTR1A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2733144-B1 NOVEL COMPOUND HAVING PARP INHIBITORY ACTIVITY SANTEN PHARMACEUTICAL CO LTD (JP) 2016-01-06 EP disclosed