SCHEMBL17429992

SCHEMBL17429992

C[C@H]1CC[C@@H](CCO)CC1

nearest known ligand 0.42

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ESR2 Q92731 2/20 0.42
BRD4 O60885 1/20 0.34
LMNA P02545 1/20 0.32
MAPK1 P28482 1/20 0.32
HTT P42858 1/20 0.32
HRH1 P35367 1/20 0.32
EPHX2 P34913 1/20 0.30
PHGDH O43175 1/20 0.30
MGLL Q99685 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2702409 1.00 ESR2 (0.42) ESR2BRD4LMNAMAPK1HTT
SCHEMBL13223460 1.00 ESR2 (0.42) ESR2BRD4LMNAMAPK1HTT
SCHEMBL14555105 0.93 ESR2 (0.38) ESR2BRD4
SCHEMBL24197652 0.85 ESR2 (0.50) ESR2BRD4
SCHEMBL240852 0.85 ESR2 (0.50) ESR2BRD4
SCHEMBL5733 0.85
SCHEMBL7865334 0.84 LMNA (0.38) ESR2LMNAMAPK1HTTHRH1
SCHEMBL12454240 0.84
SCHEMBL17133476 0.84
SCHEMBL18090623 0.84 LMNA (0.38) ESR2LMNAMAPK1HTTHRH1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9682993-B2 Anticancer compounds ST. JUDE CHILDREN'S RESEARCH HOSPITAL (US) 2017-06-20 US disclosed
US-9550741-B2 Benzoisothiazole compounds and methods of treating schizophrenia SHANGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2017-01-24 US disclosed
US-20160096811-A1 BENZOISOTHIAZOLE COMPOUNDS AND USE IN PREPARATION OF ANTIPSYCHOTIC DRUGS SHANAGHAI INSTITUTE OF PHARMACEUTICAL INDUSTRY (CN) 2016-04-07 US disclosed
US-20160009728-A1 ANTICANCER COMPOUNDS ST. JUDE CHILDREN'S RESEARCH HOSPITAL 2016-01-14 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160096811-A1 BENZOISOTHIAZOLE COMPOUNDS AND USE IN PREPARATION OF ANTIPSYCHOTIC DRUGS HTR3A, SLC6A3, HTR5A ESR2 3179/4885BRD4 1053/4885LMNA 3956/4885
US-20160009728-A1 ANTICANCER COMPOUNDS MKI67, TP53, BAX ESR2 2730/4885BRD4 1391/4885LMNA 1305/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.