SCHEMBL17447405

SCHEMBL17447405

COC(=O)/C=C/CNC(=O)c1n[nH]c2ccc(OC)cc12

nearest known ligand 0.57

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
GSK3B P49841 15/20 0.57
SMN1; SMN2 Q16637 1/20 0.52
ROCK1 Q13464 1/20 0.50
CDK2 P24941 2/20 0.49
CDK16 Q00536 1/20 0.49
DYRK1A Q13627 1/20 0.49
ROCK2 O75116 1/20 0.48
FLT3 P36888 1/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17438030 0.79 NR4A2 (0.58)
SCHEMBL17447387 0.78 ALDH1A1 (0.54)
SCHEMBL4794844 0.75 KDM4E (0.63) GSK3BSMN1; SMN2ROCK1CDK2FLT3
SCHEMBL17447381 0.74 MAPT (0.56) ROCK1ROCK2
SCHEMBL15210880 0.74 GSK3B (0.78) GSK3BCDK2CDK16DYRK1A
SCHEMBL929332 0.74 PRKAG1 (0.79) GSK3BROCK1CDK2FLT3
SCHEMBL17324787 0.74 PRKAG1 (0.62) GSK3BSMN1; SMN2ROCK1CDK2DYRK1A
SCHEMBL18910657 0.73 TUBB1 (0.50)
Hydrochloric Acid SCHEMBL15210531 0.73 GSK3B (0.76) GSK3BCDK2CDK16DYRK1A
SCHEMBL17447428 0.73 PKM (0.66) SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-10273208-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NORTHWESTERN UNIVERSITY (US) 2019-04-30 US disclosed
US-20170152228-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NORTHWESTERN UNIVERSITY (US) 2017-06-01 US disclosed
US-9586890-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NORTHWESTERN UNIVERSITY (US) 2017-03-07 US disclosed
US-20160016893-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NORTHWESTERN UNIVERSITY (US) 2016-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (3 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170152228-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NEDD4, STUB1, CUL1 GSK3B 1843/4885SMN1; SMN2 4028/4885ROCK1 1348/4885
US-20160016893-A1 SCREENING METHODS FOR THE BINDING AFFINITY OF CHEMICAL ENTITIES TO BIOLOGICAL MOLECULES AND NEDD4-1 INHIBITORS IDENTIFIED BY THE SCREENING METHODS NEDD4, STUB1, UBQLN1 GSK3B 555/4885SMN1; SMN2 2107/4885ROCK1 1815/4885
US-10273208-B2 Screening methods for the binding affinity of chemical entities to biological molecules and NEDD4-1 inhibitors identified by the screening methods NEDD4, STUB1, CUL1 GSK3B 1843/4885SMN1; SMN2 4028/4885ROCK1 1348/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.