SCHEMBL17454404

SCHEMBL17454404

CC(=O)c1cnn2cc(OCc3ccccc3)ccc12

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAOB P27338 3/20 0.54
P4HTM Q9NXG6 1/20 0.47
ALKBH1 Q13686 4/20 0.46
EPHB3 P54753 1/20 0.46
SRD5A2 P31213 1/20 0.45
SMN1; SMN2 Q16637 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.45
ALDH1A1 P00352 1/20 0.45
HTT P42858 1/20 0.45
NR4A1 P22736 1/20 0.44
NR4A2 P43354 1/20 0.44
NR4A3 Q92570 1/20 0.44
ALOX5 P09917 1/20 0.44
PTGS1 P23219 1/20 0.44
PTGS2 P35354 1/20 0.44
MAPT P10636 1/20 0.43
CYP2C9 P11712 1/20 0.43
CYP2C19 P33261 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
PLA2G4B P0C869 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17437917 0.91 ALKBH1 (0.53) MAOBP4HTMALKBH1EPHB3SRD5A2
SCHEMBL1324201 0.89 EPHB3 (0.46) MAOBP4HTMALKBH1EPHB3SRD5A2
SCHEMBL19902366 0.89 MAPT (0.46) MAOBP4HTMALKBH1EPHB3SRD5A2
SCHEMBL17452634 0.88 ALKBH1 (0.43) MAOBP4HTMALKBH1EPHB3SRD5A2
SCHEMBL3611334 0.82 EPHB3 (0.66) MAOBALKBH1EPHB3SRD5A2NR4A2
SCHEMBL17454476 0.79 LMNA (0.49) EPHB3SMN1; SMN2ALDH1A1HTTMAPT
SCHEMBL31416740 0.79 RAB9A (0.43) MAOBP4HTMALKBH1SMN1; SMN2L3MBTL1
SCHEMBL17454506 0.78 ROCK2 (0.48) EPHB3SMN1; SMN2ALDH1A1MAPT
SCHEMBL17324670 0.78 ROCK2 (0.47)
SCHEMBL17323234 0.78 LCK (0.46) EPHB3SMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20160016914-A1 SPIROCYCLOHEPTANES AS INHIBITORS OF ROCK BRISTOL-MYERS SQUIBB COMPANY 2016-01-21 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160016914-A1 SPIROCYCLOHEPTANES AS INHIBITORS OF ROCK ROCK1, MYLK, ROCK2 MAOB 2525/4885P4HTM 3285/4885ALKBH1 3389/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.