SCHEMBL1746128

SCHEMBL1746128

Cc1cc2cnn(CCO[Si](C)(C)C(C)(C)C)c2cc1N.Cc1cc2cnn(CCO[Si](C)(C)C(C)(C)C)c2cc1[N+](=O)[O-]

nearest known ligand 0.36

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
GLS O94925 1/20 0.34
GAA P10253 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP3A4 P08684 1/20 0.32
TSHR P16473 1/20 0.32
RECQL P46063 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1464500 0.94 GLS (0.38) GLSGAAALDH1A1CYP3A4TSHR
SCHEMBL1746766 0.89 HTR2A (0.32)
SCHEMBL1463344 0.89 HTR2A (0.32)
SCHEMBL1746159 0.85 GLS (0.32) GLSALDH1A1CYP3A4
SCHEMBL1744945 0.82 DUT (0.36) GAAALDH1A1CYP3A4TSHRRECQL
Hydrazinecarboxamide SCHEMBL1464009 0.82 KMO (0.36)
SCHEMBL31716743 0.79 GLS (0.42) GLSGAAALDH1A1CYP3A4TSHR
SCHEMBL16931512 0.76 GLS (0.61) GLSALDH1A1
SCHEMBL1744241 0.75 DUT (0.40) ALDH1A1
SCHEMBL16899218 0.72 KMT2A (0.35) GAAALDH1A1CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2385939-A1 DIHYDROPYRIDONE AMIDES AS P2X7 MODULATORS F. Hoffmann-La Roche AG (CH) 2011-11-16 EP disclosed
US-8041551-B1 Algorithm and architecture for multi-argument associative operations that minimizes the number of components using a latency of the components THE MATHWORKS, INC. (US) 2011-10-18 US disclosed
WO-2010072597-A1 DIHYDROPYRIDONE AMIDES AS P2X7 MODULATORS F. HOFFMANN-LA ROCHE AG (CH) 2010-07-01 WO disclosed