SCHEMBL17469286

SCHEMBL17469286

COc1cc(OCC(F)(F)F)c2[nH]c(C(F)(F)F)c(C(=O)C(F)(F)F)c2c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
BCHE P06276 1/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C9 P11712 1/20 0.36
NQO2 P16083 1/20 0.35
ALDH1A1 P00352 2/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
KDM4E B2RXH2 1/20 0.33
CYP3A4 P08684 1/20 0.32
HPGD P15428 1/20 0.32
CYP2C19 P33261 1/20 0.32
ATM Q13315 1/20 0.32
POLB P06746 1/20 0.32
MTNR1A P48039 1/20 0.32
MTNR1B P49286 1/20 0.32
TRPV1 Q8NER1 1/20 0.32
ELANE P08246 1/20 0.31
DYRK1A Q13627 1/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17469282 0.89 NQO2 (0.45) BCHENQO2KDM4ECYP3A4HPGD
SCHEMBL17469274 0.82 CYP3A4 (0.38) BCHENQO2ALDH1A1MEN1KMT2A
SCHEMBL17469285 0.82 CFTR (0.41) BCHENQO2ALDH1A1MEN1KMT2A
SCHEMBL17469279 0.82 ENPP3 (0.38) BCHENQO2MEN1KMT2AKDM4E
SCHEMBL17469275 0.81 BCHE (0.36) BCHECYP1A2NQO2CYP3A4CYP2C19
SCHEMBL17469281 0.81 BCHE (0.36) BCHENQO2MEN1KMT2AKDM4E
SCHEMBL19322129 0.79 GAA (0.40) BCHECYP1A2CYP2C9ALDH1A1MEN1
SCHEMBL17469284 0.78 PDE3B (0.39) CYP1A2CYP2C9ALDH1A1MEN1KMT2A
SCHEMBL19317480 0.77 PDE3B (0.36) CYP1A2CYP2C9NQO2ALDH1A1MEN1
SCHEMBL19317478 0.76 ALOX5 (0.36) CYP1A2CYP2C9ALDH1A1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-11147795-B2 Neuroprotective compounds and methods of use ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2021-10-19 US disclosed
US-20190350902-A1 NEUROPROTECTIVE COMPOUNDS AND METHODS OF USE ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2019-11-21 US disclosed
US-10358438-B2 [3+2] annulation to produce 5-membered heterocyclic compounds ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2019-07-23 US disclosed
US-20170253580-A1 ORGANIC REACTIONS THE ARIZONA BOARD OF REGENTS ON BEHALF OF THE UNIVERSITY OF ARIZONA (US) 2017-09-07 US disclosed
WO-2016014426-A1 ORGANIC REACTIONS THE ARIZONA BOARD OF REGENTS (US) 2016-01-28 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (4 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-11147795-B2 Neuroprotective compounds and methods of use RTN3, CHRNB3, ARRB1 BCHE 1054/4885CYP1A2 1866/4885CYP2C9 3689/4885
US-20170253580-A1 ORGANIC REACTIONS MYC, CYP2E1, CYP3A4 BCHE 1609/4885CYP1A2 28/4885CYP2C9 32/4885
US-20190350902-A1 NEUROPROTECTIVE COMPOUNDS AND METHODS OF USE RTN3, CHRNB3, ARRB1 BCHE 1054/4885CYP1A2 1866/4885CYP2C9 3689/4885
US-10358438-B2 [3+2] annulation to produce 5-membered heterocyclic compounds ACR, MYC, TOP1 BCHE 2514/4885CYP1A2 45/4885CYP2C9 77/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.