SCHEMBL174763

SCHEMBL174763

Cc1nn(C)c(-c2ccc(F)cc2Cl)c1NC(=O)O

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
P2RX7 Q99572 4/20 0.45
CYP1A2 P05177 2/20 0.43
CYP2C19 P33261 2/20 0.43
SCN10A Q9Y5Y9 1/20 0.43
HSD11B1 P28845 1/20 0.42
LMNA P02545 2/20 0.41
ALDH1A1 P00352 1/20 0.41
SMN1; SMN2 Q16637 1/20 0.41
MAPT P10636 1/20 0.41
NR3C1 P04150 1/20 0.41
GRM5 P41594 3/20 0.40
IGF1R P08069 1/20 0.40
CYP3A4 P08684 3/20 0.40
CYP2C9 P11712 1/20 0.40
GRM2 Q14416 1/20 0.39
HTT P42858 1/20 0.39
POLB P06746 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL173927 0.89 CYP1A2 (0.48) P2RX7CYP1A2CYP2C19SCN10AHSD11B1
SCHEMBL174691 0.83 P2RX7 (0.43) P2RX7CYP1A2CYP2C19SCN10AHSD11B1
SCHEMBL174040 0.81 MAPK1 (0.45) P2RX7HSD11B1IGF1R
SCHEMBL175155 0.80 ALDH1A1 (0.44) P2RX7CYP1A2CYP2C19SCN10AHSD11B1
SCHEMBL20673409 0.79 CYP1A2 (0.46) P2RX7CYP1A2CYP2C19SCN10AHSD11B1
SCHEMBL173503 0.77 HSD11B1 (0.47) P2RX7SCN10AHSD11B1IGF1RGRM2
SCHEMBL14990088 0.77 CYP1A2 (0.42) CYP1A2CYP2C19HSD11B1IGF1RCYP3A4
SCHEMBL175196 0.77 CRHR1 (0.42) CYP1A2CYP2C19HSD11B1IGF1RCYP3A4
SCHEMBL175200 0.77 HSD11B1 (0.40) P2RX7CYP1A2CYP2C19HSD11B1IGF1R
SCHEMBL174924 0.74 LMNA (0.54) P2RX7HSD11B1LMNAALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9131693-B2 Fungicidal pyrazoles E I DU PONT DE NEMOURS AND COMPANY (US) 2015-09-15 US disclosed
EP-2611297-B1 FUNGICIDAL PYRAZOLES DU PONT (US) 2015-06-17 EP disclosed
US-20140221448-A1 FUNGICIDAL PYRAZOLES E I DU PONT DE NEMOURS AND COMPANY (US) 2014-08-07 US disclosed
US-8754115-B2 Fungicidal pyrazoles E I DU PONT DE NEMOURS AND COMPANY (US) 2014-06-17 US disclosed
EP-2611297-A1 FUNGICIDAL PYRAZOLES E.I. Du Pont De Nemours And Company (US) 2013-07-10 EP disclosed
US-20130143940-A1 FUNGICIDAL PYRAZOLES E I DU PONT DE NEMOURS AND COMPANY (US) 2013-06-06 US disclosed
WO-2012030922-A1 FUNGICIDAL PYRAZOLES E. I. DU PONT DE NEMOURS AND COMPANY (US) 2012-03-08 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20140221448-A1 FUNGICIDAL PYRAZOLES CYP1A1, CYP1B1, CYP4X1 P2RX7 316/4885CYP1A2 8/4885CYP2C19 43/4885
US-20130143940-A1 FUNGICIDAL PYRAZOLES CYP1A1, CYP1B1, CYP4X1 P2RX7 316/4885CYP1A2 8/4885CYP2C19 43/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.