SCHEMBL17478588

SCHEMBL17478588

O=C(c1ccccc1)[C@]1(C(=O)c2ccc(Br)cc2)C[C@H](O)CN1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MAPT P10636 4/20 0.38
AKR1C3 P42330 1/20 0.36
MEN1 O00255 3/20 0.36
KMT2A Q03164 3/20 0.36
NPC1 O15118 3/20 0.36
RAB9A P51151 3/20 0.36
TP53 P04637 1/20 0.36
HPGD P15428 1/20 0.36
SMN1; SMN2 Q16637 3/20 0.35
KDM4E B2RXH2 2/20 0.35
ESRRG P62508 1/20 0.35
F2RL1 P55085 1/20 0.35
CYP1B1 Q16678 1/20 0.35
CYP3A4 P08684 2/20 0.35
CYP1A2 P05177 1/20 0.35
NFKB1 P19838 1/20 0.35
CYP2C19 P33261 1/20 0.35
CASP3 P42574 1/20 0.35
NFKB2 Q00653 1/20 0.35
RELA Q04206 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17478610 1.00 MAPT (0.38) MAPTAKR1C3MEN1KMT2ANPC1
SCHEMBL17478651 0.91 LMNA (0.37) CYP2C19CES2CES1ALDH1A1LMNA
SCHEMBL17478616 0.91 LMNA (0.37) CYP2C19CES2CES1ALDH1A1LMNA
SCHEMBL5654938 0.66 ARG1 (0.45) MAPTMEN1KMT2ANPC1RAB9A
SCHEMBL10415978 0.65 MAPT (0.41) MAPTAKR1C3MEN1KMT2ANPC1
SCHEMBL10414509 0.65 LMNA (0.43) MAPTAKR1C3MEN1KMT2ANPC1
SCHEMBL649996 0.64 CES2 (0.80) MAPTAKR1C3MEN1KMT2ANPC1
Benzophenone SCHEMBL11774383 0.64 ALDH1A1 (0.70) MAPTAKR1C3MEN1KMT2ANPC1
Benzoic Acid SCHEMBL28594970 0.64 TSHR (0.70) MAPTAKR1C3MEN1KMT2ANPC1
SCHEMBL69395 0.64 ALDH1A1 (0.70) MAPTAKR1C3MEN1KMT2ANPC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3174886-A1 2-OXA-5-AZABICYCLO[2.2.1]HEPTAN-3-YL DERIVATIVES F. Hoffmann-La Roche AG (CH) 2017-06-07 EP disclosed
WO-2016016292-A1 2-OXA-5-AZABICYCLO[2.2.1]HEPTAN-3-YL DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2016-02-04 WO disclosed
WO-2016015333-A1 2-OXA-5-AZABICYCLO [2.2.1] HEPTAN-3-YL DERIVATIVES F.HOFFMANN-LA ROCHE AG (CH) 2016-02-04 WO disclosed