SCHEMBL17495183

SCHEMBL17495183

CCSc1cc(Br)ccc1C(=O)O

nearest known ligand 0.57

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PTPRC P08575 1/20 0.57
PTPRG P23470 1/20 0.57
KDM4E B2RXH2 2/20 0.44
GLA P06280 1/20 0.44
POLB P06746 2/20 0.42
MYC P01106 1/20 0.41
NR4A1 P22736 1/20 0.41
RXFP1 Q9HBX9 3/20 0.41
TSHR P16473 1/20 0.40
HSD17B10 Q99714 1/20 0.40
APEX1 P27695 1/20 0.40
MEN1 O00255 2/20 0.39
KMT2A Q03164 2/20 0.39
CYP1A2 P05177 2/20 0.39
SORT1 Q99523 2/20 0.38
PRNP P04156 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
PPARG P37231 1/20 0.38
HIF1A Q16665 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL30969147 0.86 PTPRC (0.43) PTPRCPTPRGTSHRCYP1A2CYP2C9
SCHEMBL17732190 0.86 PTPRC (0.43) PTPRCPTPRGTSHRCYP1A2CYP2C9
SCHEMBL20482053 0.85 PTPRC (0.46) PTPRCPTPRGKDM4EGLAPOLB
SCHEMBL17494851 0.82 NR4A2 (0.46) PTPRCPTPRGKDM4EGLAPOLB
SCHEMBL28229958 0.82 PTPRC (0.53) PTPRCPTPRGKDM4EGLAPOLB
SCHEMBL4611677 0.81 ALDH1A1 (0.49) KDM4ERXFP1TSHRHSD17B10MEN1
SCHEMBL20152377 0.81 CSNK2A1 (0.47) PTPRCPTPRGKDM4EPOLBMEN1
SCHEMBL3198739 0.80 PTPRC (0.50) PTPRCPTPRGKDM4EGLAPOLB
SCHEMBL9952116 0.79 KEAP1 (0.44) PTPRCPTPRGKDM4EPOLBHSD17B10
SCHEMBL20505156 0.79 PTPRC (0.53) PTPRCPTPRGKDM4EGLAPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 37 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3802542-B1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULFOXIMINE CONTAINING SUBSTITUENTS SYNGENTA CROP PROTECTION AG (CH) 2025-05-28 EP disclosed
CN-119431377-A Pesticidally active heterocyclic derivatives with sulfoximine containing substituents 先正达农作物保护股份公司 2025-02-14 CN disclosed
CN-112262140-B Pesticidally active heterocyclic derivatives with sulfoximine containing substituents 先正达农作物保护股份公司 2024-05-28 CN disclosed
EP-4342297-A2 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULFOXIMINE CONTAINING SUBSTITUENTS Syngenta Crop Protection AG (CH) 2024-03-27 EP disclosed
US-20230150944-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULFOXIMINE CONTAINING SUBSTITUENTS SYNGENTA CROP PROTECTION AG (CH) 2023-05-18 US disclosed
EP-3180341-B1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2022-04-27 EP disclosed
EP-3180341-B1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2022-04-27 EP disclosed
EP-3802542-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULFOXIMINE CONTAINING SUBSTITUENTS Syngenta Crop Protection AG (CH) 2021-04-14 EP disclosed
CN-112262140-A Pesticidally active heterocyclic derivatives with sulfoximine-containing substituents 先正达农作物保护股份公司 2021-01-22 CN disclosed
EP-3186249-B1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2020-12-09 EP disclosed
US-20170233389-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2017-08-17 US disclosed
EP-3186249-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS Syngenta Participations AG (CH) 2017-07-05 EP disclosed
EP-3183245-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS Syngenta Participations AG (CH) 2017-06-28 EP disclosed
EP-3180341-A2 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS Syngenta Participations AG (CH) 2017-06-21 EP disclosed
WO-2016120182-A1 PESTICIDALLY ACTIVE AMIDE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2016-08-04 WO disclosed
WO-2016120182-A1 PESTICIDALLY ACTIVE AMIDE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2016-08-04 WO disclosed
WO-2016030229-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2016-03-03 WO disclosed
WO-2016026848-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2016-02-25 WO disclosed
WO-2016023954-A2 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2016-02-18 WO disclosed
WO-2016023954-A2 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS SYNGENTA PARTICIPATIONS AG (CH) 2016-02-18 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (2 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20170233389-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULPHUR CONTAINING SUBSTITUENTS DDT, ACHE, GSTM1 PTPRC 2441/4885PTPRG 1657/4885KDM4E 2839/4885
US-20230150944-A1 PESTICIDALLY ACTIVE HETEROCYCLIC DERIVATIVES WITH SULFOXIMINE CONTAINING SUBSTITUENTS AADAC, ACHE, DDT PTPRC 3587/4885PTPRG 2399/4885KDM4E 1746/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.