SCHEMBL17508271

SCHEMBL17508271

COc1ccc(-c2ccc(C=O)cc2)c(C)c1

nearest known ligand 0.58

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.58
CYP2A6 P11509 2/20 0.58
SMN1; SMN2 Q16637 1/20 0.45
KDM4E B2RXH2 1/20 0.44
CYP1A2 P05177 1/20 0.44
CYP2D6 P10635 1/20 0.44
CYP2C9 P11712 1/20 0.44
CYP2C19 P33261 1/20 0.44
PTGER4 P35408 1/20 0.42
ERN1 O75460 2/20 0.41
TRIM24 O15164 1/20 0.41
TYR P14679 1/20 0.41
TRIM33 Q9UPN9 1/20 0.41
GSTP1 P09211 1/20 0.41
DRD1 P21728 1/20 0.41
TUBB1 Q9H4B7 1/20 0.41
ALDH1A3 P47895 1/20 0.41
TSHR P16473 1/20 0.41
MAOB P27338 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL31374896 1.00 ALDH1A1 (0.58) ALDH1A1CYP2A6SMN1; SMN2KDM4ECYP1A2
SCHEMBL679848 0.84 SMN1; SMN2 (0.55) CYP2A6SMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL9135095 0.83 SMN1; SMN2 (0.41) CYP2A6SMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL12740233 0.83 ERN1 (0.58) ALDH1A1CYP2A6SMN1; SMN2CYP1A2CYP2D6
SCHEMBL17508246 0.82 ERN1 (0.57) ALDH1A1CYP2A6SMN1; SMN2KDM4ECYP1A2
SCHEMBL2014355 0.82 ALDH1A1 (0.56) ALDH1A1CYP2A6SMN1; SMN2KDM4ECYP1A2
SCHEMBL4455043 0.81 KDM4E (0.45) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL10068337 0.80 ACHE (0.54) ALDH1A1SMN1; SMN2KDM4ECYP1A2CYP2D6
SCHEMBL26628327 0.80 ALDH1A1 (0.58) ALDH1A1CYP2A6KDM4EERN1TRIM24
SCHEMBL4896568 0.80 ALDH1A1 (0.50) ALDH1A1CYP2A6SMN1; SMN2KDM4ECYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed
WO-2016019588-A1 OXACAZONE COMPOUNDS TO TREAT CLOSTRIDIUM DIFFICILE THE BROAD INSTITUTE, INC. (US) 2016-02-11 WO disclosed