SCHEMBL17524934

SCHEMBL17524934

O=C1Nc2ncccc2C12CCN(c1cnc(Br)cn1)CC2

nearest known ligand 0.39

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CALCA P06881 5/20 0.39
CALCRL Q16602 11/20 0.34
PTPN11 Q06124 2/20 0.34
ADRA2B P18089 1/20 0.34
OTUD7B Q6GQQ9 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524906 0.87 CALCA (0.40) CALCACALCRLPTPN11
SCHEMBL17506417 0.82 CALCA (0.40) CALCACALCRL
SCHEMBL17524992 0.81 CALCA (0.39) CALCAOTUD7B
SCHEMBL17524937 0.81 ME2 (0.40) CALCACALCRL
SCHEMBL17524949 0.77 CALCA (0.41) CALCACALCRLOTUD7B
SCHEMBL13806581 0.77 CALCA (0.46) CALCACALCRLOTUD7B
SCHEMBL16235885 0.76 CALCA (0.46) CALCACALCRLOTUD7B
SCHEMBL12655392 0.76 CALCA (0.47) CALCACALCRLOTUD7B
SCHEMBL1700112 0.76 CALCA (0.49) CALCACALCRLOTUD7B
SCHEMBL12400699 0.76 CALCA (0.45) CALCACALCRLOTUD7B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed