SCHEMBL17524992

SCHEMBL17524992

Cc1ccc(N2CCC3(CC2)C(=O)Nc2ncccc23)nc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CALCA P06881 3/20 0.39
GRIN2D O15399 1/20 0.39
GRIN3B O60391 1/20 0.39
GRIN1 Q05586 1/20 0.39
GRIN2A Q12879 1/20 0.39
GRIN2B Q13224 1/20 0.39
GRIN2C Q14957 1/20 0.39
GRIN3A Q8TCU5 1/20 0.39
CRBN Q96SW2 4/20 0.38
OTUD7B Q6GQQ9 1/20 0.38
NPC1 O15118 1/20 0.38
ALDH1A1 P00352 1/20 0.38
CYP1A2 P05177 1/20 0.38
GAA P10253 1/20 0.38
MAPT P10636 1/20 0.38
CYP2C9 P11712 1/20 0.38
CYP2C19 P33261 1/20 0.38
RAB9A P51151 1/20 0.38
MCL1 Q07820 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524906 0.87 CALCA (0.40) CALCAHTR7KCNH2
SCHEMBL17506417 0.87 CALCA (0.40) CALCAGRIN2DGRIN3BGRIN1GRIN2A
SCHEMBL17524937 0.86 ME2 (0.40) CALCACRBNKCNH2
SCHEMBL17525083 0.84 CRBN (0.40) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL17525112 0.82 SCN9A (0.43) CALCACRBNCYP2C9SCN9A
SCHEMBL17525014 0.82 CALCA (0.38) CALCACRBNKCNH2
SCHEMBL17524934 0.81 CALCA (0.39) CALCAOTUD7B
SCHEMBL17524991 0.80 DRD2 (0.38) GRIN2DGRIN3BGRIN1GRIN2AGRIN2B
SCHEMBL17524997 0.80 EGLN1 (0.43) CALCAHTR7KCNH2
SCHEMBL1700112 0.79 CALCA (0.49) CALCAOTUD7B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed