SCHEMBL17525083

SCHEMBL17525083

Cc1ccc(N2CCC3(CC2)C(=O)Nc2ncncc23)nc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CRBN Q96SW2 6/20 0.40
DDB1 Q16531 2/20 0.37
LCAT P04180 1/20 0.37
GRIN2D O15399 1/20 0.36
GRIN3B O60391 1/20 0.36
GRIN1 Q05586 1/20 0.36
GRIN2A Q12879 1/20 0.36
GRIN2B Q13224 1/20 0.36
GRIN2C Q14957 1/20 0.36
GRIN3A Q8TCU5 1/20 0.36
GPR119 Q8TDV5 2/20 0.36
DHFR P00374 1/20 0.36
SCN9A Q15858 2/20 0.36
BPTF Q12830 1/20 0.36
DRD2 P14416 3/20 0.35
DRD1 P21728 3/20 0.35
DRD5 P21918 3/20 0.35
DRD3 P35462 3/20 0.35
HTR1A P08908 1/20 0.35
DRD4 P21917 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17524992 0.84 CALCA (0.39) CRBNLCATGRIN2DGRIN3BGRIN1
SCHEMBL17524991 0.80 DRD2 (0.38) CRBNLCATGRIN2DGRIN3BGRIN1
SCHEMBL15935920 0.79 FGFR1 (0.38)
SCHEMBL29388502 0.76 MAP3K11 (0.39)
SCHEMBL30748859 0.74 MAP3K11 (0.43)
SCHEMBL30748975 0.74 MAP3K11 (0.46)
SCHEMBL17525060 0.73 MAPT (0.39)
SCHEMBL30749023 0.72 MAP3K11 (0.45)
SCHEMBL15935911 0.72 CALCRL (0.39)
SCHEMBL13748469 0.71 BACE1 (0.36)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016022644-A1 HETEROCYCLIC CGRP RECEPTOR ANTAGONISTS MERCK SHARP & DOHME CORP. (US) 2016-02-11 WO disclosed