SCHEMBL17525967

SCHEMBL17525967

C[C@@]12CCCC1C1CCc3c(ccc(C#N)c3F)C1CC2

nearest known ligand 0.53

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
SHBG P04278 1/20 0.53
STS P08842 8/20 0.47
CYP19A1 P11511 2/20 0.47
ESR1 P03372 3/20 0.39
ESR2 Q92731 3/20 0.39
KDM4E B2RXH2 1/20 0.39
MEN1 O00255 1/20 0.39
LMNA P02545 1/20 0.39
GAA P10253 1/20 0.39
MAPT P10636 1/20 0.39
G6PD P11413 1/20 0.39
PKM P14618 1/20 0.39
MAPK1 P28482 1/20 0.39
MPI P34949 1/20 0.39
KMT2A Q03164 1/20 0.39
HSD17B1 P14061 2/20 0.38
MBOAT4 Q96T53 2/20 0.36
ABCB11 O95342 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL14048707 0.97 SHBG (0.49) SHBGSTSCYP19A1ESR1ESR2
SCHEMBL14048673 0.84 SHBG (0.50) SHBGSTSCYP19A1ESR1ESR2
SCHEMBL14048674 0.83 SHBG (0.52) SHBGSTSCYP19A1ESR1ESR2
SCHEMBL13951923 0.81 STS (0.72) SHBGSTSCYP19A1ESR1ESR2
SCHEMBL13952155 0.78 STS (0.46) STSCYP19A1ESR1ESR2KDM4E
SCHEMBL17525951 0.78 CYP19A1 (0.53) STSCYP19A1ESR1ESR2KDM4E
SCHEMBL7596151 0.77 SHBG (0.58) SHBGSTSCYP19A1ESR1ESR2
SCHEMBL17525944 0.75 SHBG (0.70) SHBGSTSCYP19A1ESR1ESR2
SCHEMBL13952148 0.74 STS (0.56) SHBGSTSCYP19A1ESR1ESR2
SCHEMBL13952156 0.74 STS (0.56) SHBGSTSCYP19A1ESR1ESR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-2147014-B1 17ALPHA-SUBSTITUTED STEROIDS AS SYSTEMIC ANTIANDROGENS AND SELECTIVE ANDROGEN RECEPTOR MODULATORS ENDORECH INC (CA) 2016-02-17 EP disclosed