SCHEMBL17529971

SCHEMBL17529971

CC(C)CC(NC(=O)N1CCCC(c2ccccc2)C1)C(=O)NCC#N

nearest known ligand 0.56

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
CTSS P25774 10/20 0.56
CTSL P07711 8/20 0.54
CTSK P43235 5/20 0.54
CTSB P07858 3/20 0.54
HSD11B1 P28845 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17530239 0.91 CTSL (0.56) CTSSCTSLCTSKCTSB
SCHEMBL17530013 0.90 CTSL (0.56) CTSSCTSLCTSKCTSB
SCHEMBL17530194 0.90 CTSS (0.52) CTSSCTSLCTSKCTSBHSD11B1
SCHEMBL17530227 0.89 HSD11B1 (0.46) CTSSCTSLCTSKCTSBHSD11B1
SCHEMBL17530170 0.89 CTSS (0.51) CTSSCTSLCTSKCTSB
SCHEMBL17529976 0.89 CTSS (0.62) CTSSCTSLCTSKCTSB
SCHEMBL17530199 0.88 CTSS (0.48) CTSSCTSLCTSKCTSB
SCHEMBL17530402 0.88 CTSS (0.52) CTSSCTSLCTSKCTSB
SCHEMBL17530189 0.86 CTSS (0.46) CTSSCTSLCTSKCTSB
SCHEMBL17529998 0.86 CTSS (0.50) CTSSCTSLCTSKCTSB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016027284-A2 PIPERIDINE UREAS AS CATHEPSIN CYSTEINE PROTEASE INHIBITORS ALKEM LABORATORIES LTD. (IN) 2016-02-25 WO disclosed