SCHEMBL17530362

SCHEMBL17530362

CC(C)(F)CC(NC(=O)N1CCC(c2ccccc2)CC1)C(N)=O

nearest known ligand 0.53

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.46
HSD11B1 P28845 1/20 0.45
KCNH2 Q12809 1/20 0.44
HRH3 Q9Y5N1 1/20 0.44
CHRM4 P08173 1/20 0.44
GAA P10253 1/20 0.44
CCR1 P32246 5/20 0.43
POLB P06746 1/20 0.43
NAMPT P43490 1/20 0.43
TP53 P04637 1/20 0.43
RAB9A P51151 1/20 0.43
SMN1; SMN2 Q16637 1/20 0.43
CHRM2 P08172 1/20 0.42
CHRM5 P08912 1/20 0.42
CHRM1 P11229 1/20 0.42
CHRM3 P20309 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17530209 0.91 CCR1 (0.47) NPC1CHRM4CCR1POLBNAMPT
SCHEMBL17530392 0.84 CTSL (0.53) NPC1CHRM4POLB
SCHEMBL17530364 0.80 CTSB (0.64)
SCHEMBL17530360 0.78 ROCK2 (0.46) GAA
SCHEMBL17529990 0.77 CTSL (0.60) CHRM4CCR1
SCHEMBL10122318 0.74 NPC1 (0.52) NPC1HSD11B1KCNH2HRH3CHRM4
SCHEMBL10123588 0.72 NPC1 (0.50) NPC1HSD11B1KCNH2HRH3CHRM4
SCHEMBL18560441 0.71 PSMB11 (0.47) NPC1CHRM4GAACCR1POLB
SCHEMBL12320990 0.70 MMP3 (0.50) NPC1HSD11B1GAACCR1POLB
SCHEMBL12321693 0.70 MMP3 (0.50) NPC1HSD11B1GAACCR1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016027284-A2 PIPERIDINE UREAS AS CATHEPSIN CYSTEINE PROTEASE INHIBITORS ALKEM LABORATORIES LTD. (IN) 2016-02-25 WO disclosed