SCHEMBL175591

SCHEMBL175591

CC(=O)OCCc1ccc(C(=O)c2sc(N)nc2-c2cccc(C#N)c2)cc1

nearest known ligand 0.47

Predicted protein targets (top 11)

geneUniProtsupporting neighboursconfidence
RORC P51449 2/20 0.47
ALDH1A1 P00352 1/20 0.40
HSD17B10 Q99714 1/20 0.40
KDM1A O60341 1/20 0.40
RORB Q92753 9/20 0.39
VNN1 O95497 2/20 0.36
MMP12 P39900 1/20 0.36
MMP13 P45452 1/20 0.36
ADORA2A P29274 2/20 0.35
ADORA1 P30542 2/20 0.35
ADORA3 P0DMS8 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL176165 0.85 ALDH1A1 (0.55) ALDH1A1HSD17B10RORBADORA2AADORA1
SCHEMBL175366 0.82 ALDH1A1 (0.53) ALDH1A1HSD17B10RORBADORA2AADORA1
SCHEMBL175512 0.81 RORB (0.54) RORCALDH1A1HSD17B10RORBADORA2A
SCHEMBL6288104 0.76 ALDH1A1 (0.69) ALDH1A1HSD17B10ADORA2A
SCHEMBL174906 0.72 RORB (0.74) RORCRORBADORA2AADORA1
SCHEMBL4267596 0.70 ALDH1A1 (0.55) RORCALDH1A1HSD17B10RORBADORA2A
SCHEMBL175193 0.70 ALDH1A1 (0.52) RORCALDH1A1HSD17B10RORBADORA2A
SCHEMBL17316360 0.68 KDM1A (0.50) ALDH1A1HSD17B10KDM1AMMP12MMP13
SCHEMBL1256197 0.68 ADORA2A (0.49) ALDH1A1HSD17B10ADORA2AADORA1ADORA3
SCHEMBL10092885 0.67 RORB (0.70) RORCRORBADORA2AADORA1ADORA3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed
WO-2012027965-A1 NOVEL COMPOUNDS GLAXO GROUP LIMITED (GB) 2012-03-08 WO disclosed