SCHEMBL1758703

SCHEMBL1758703

O=C(Cc1csc(N(CC23CC4CC(C2)CC(c2ccccc2)(C4)C3)C(=O)O)n1)NO

nearest known ligand 0.57

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PDE5A O76074 8/20 0.40
KDM4E B2RXH2 1/20 0.40
PDE1A P54750 3/20 0.39
PDE1B Q01064 3/20 0.39
PDE1C Q14123 3/20 0.39
SPHK2 Q9NRA0 1/20 0.38
LMNA P02545 1/20 0.37
MEN1 O00255 1/20 0.36
KMT2A Q03164 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1758697 0.85 PDE5A (0.40) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758601 0.80 PDE5A (0.54) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758738 0.79 PDE5A (0.48) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758679 0.78 PDE5A (0.41) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758880 0.77 PDE5A (0.41) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758740 0.77 PDE5A (0.37) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758935 0.76 PDE5A (0.39) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758817 0.75 PDE5A (0.50) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758659 0.70 PDE5A (0.38) PDE5AKDM4EPDE1APDE1BPDE1C
SCHEMBL1758680 0.69 ALDH1A1 (0.42) PDE5AKDM4EPDE1APDE1BPDE1C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2011058582-A1 HISTONE DEACETYLASE INHIBITORS FOR THE TREATMENT OF FUNGAL INFECTIONS ORCHID RESEARCH LABORATORIES LTD. (IN) 2011-05-19 WO disclosed