SCHEMBL17595374

SCHEMBL17595374

CCc1cc(C(=O)OC(=O)c2c(O)c(CC)c(-c3cnn(C)c3)[nH]c2=O)c(=O)[nH]c1-c1cnn(C)c1

nearest known ligand 0.33

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AURKA O14965 1/20 0.33
TTK P33981 1/20 0.33
AURKB Q96GD4 1/20 0.33
INCENP Q9NQS7 1/20 0.33
CSF1R P07333 1/20 0.31
PDGFRA P16234 1/20 0.31
FLT3 P36888 1/20 0.31
EZH2 Q15910 7/20 0.31
PDE3B Q13370 1/20 0.31
PDE3A Q14432 1/20 0.31
ERN1 O75460 1/20 0.31
MAPK1 P28482 1/20 0.30
KDM4E B2RXH2 1/20 0.30
PIK3CD O00329 1/20 0.30
EED O75530 1/20 0.30
RBBP4 Q09028 1/20 0.30
SUZ12 Q15022 1/20 0.30
AEBP2 Q6ZN18 1/20 0.30
ADH5 P11766 3/20 0.30
KDM5A P29375 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17595373 0.86 AURKA (0.34) AURKATTKAURKBINCENPERN1
SCHEMBL17597598 0.84 USP7 (0.41) KDM5BBRD4
SCHEMBL14746098 0.80 AURKA (0.38) AURKATTKAURKBINCENPERN1
SCHEMBL17597694 0.80 PTGER3 (0.31) PDE3BPDE3A
SCHEMBL17594871 0.79 ALDH1A1 (0.39) EZH2PDE3BPDE3A
SCHEMBL17595195 0.79 KDM5A (0.32) PDE3BPDE3AKDM4EKDM5AKDM5B
SCHEMBL17594971 0.79 LMNA (0.39) PDE3BPDE3A
SCHEMBL14741179 0.78 CREBBP (0.40) AURKATTKAURKBINCENPMAPK1
SCHEMBL17595256 0.78 PDE3B (0.35) PDE3BPDE3AKDM4E
SCHEMBL17597217 0.77 MTNR1A (0.33) PDE3BPDE3A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed