SCHEMBL17594871

SCHEMBL17594871

CCc1cc(C(=O)OC(=O)c2c(O)c(CC)c(-c3ccc(N4CCCC4)cc3)[nH]c2=O)c(=O)[nH]c1-c1ccc(N2CCCC2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 2/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
LMNA P02545 1/20 0.38
PARP1 P09874 1/20 0.37
PARP2 Q9UGN5 1/20 0.37
SIRT2 Q8IXJ6 1/20 0.35
SIRT1 Q96EB6 1/20 0.35
KIF11 P52732 3/20 0.35
CNR2 P34972 1/20 0.35
MAPT P10636 1/20 0.35
KCNH2 Q12809 1/20 0.34
PDE3B Q13370 1/20 0.34
PDE3A Q14432 1/20 0.34
MEN1 O00255 1/20 0.33
KMT2A Q03164 1/20 0.33
HTT P42858 1/20 0.33
TLR9 Q9NR96 3/20 0.32
TLR8 Q9NR97 3/20 0.32
TLR7 Q9NYK1 3/20 0.32
EGFR P00533 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL17594971 0.99 LMNA (0.39) ALDH1A1L3MBTL1LMNAPARP1PARP2
SCHEMBL17594868 0.87 KIF11 (0.38) ALDH1A1L3MBTL1LMNAPARP1PARP2
SCHEMBL17594969 0.86 KIF11 (0.39) ALDH1A1LMNAPARP1PARP2SIRT2
SCHEMBL17595142 0.85 ABCB1 (0.39) ALDH1A1LMNAMAPTMEN1KMT2A
SCHEMBL14745803 0.82 DCTPP1 (0.40) ALDH1A1LMNAPARP1PARP2SIRT2
SCHEMBL17595256 0.82 PDE3B (0.35) ALDH1A1LMNAMAPTPDE3BPDE3A
SCHEMBL17594967 0.82 ALDH1A1 (0.37) ALDH1A1L3MBTL1LMNAPDE3BPDE3A
SCHEMBL14747044 0.81 KIF11 (0.41) ALDH1A1L3MBTL1LMNAPARP1PARP2
SCHEMBL14745564 0.80 KIF11 (0.42) ALDH1A1PARP1PARP2SIRT2SIRT1
SCHEMBL17595374 0.79 AURKA (0.33) PDE3BPDE3AEZH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2016039936-A2 MONOCYCLIC SUBSTITUTED 2-PYRIDINONE ANTIBACTERIAL COMPOUNDS PTC THERAPEUTICS, INC. (US) 2016-03-17 WO claimed